SCHEMBL1897684

SCHEMBL1897684

Nc1nc2ccccc2[nH]c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAUR Q03405 1/20 1.00
MEN1 O00255 4/20 0.64
KMT2A Q03164 4/20 0.64
RAB9A P51151 8/20 0.60
NPC1 O15118 7/20 0.60
ALDH1A1 P00352 5/20 0.59
MASP2 O00187 1/20 0.59
NUDT1 P36639 1/20 0.59
AOC3 Q16853 1/20 0.59
KDM4E B2RXH2 8/20 0.58
KHK P50053 1/20 0.56
PDGFRB P09619 2/20 0.55
FGFR1 P11362 2/20 0.55
KDR P35968 2/20 0.55
CHEK1 O14757 1/20 0.55
FLT1 P17948 1/20 0.55
HTT P42858 4/20 0.53
HSD17B10 Q99714 3/20 0.53
HPGD P15428 2/20 0.53
GAA P10253 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30682553 1.00 PLAUR (1.00) PLAURMEN1KMT2ARAB9ANPC1
SCHEMBL30588935 0.79 KMT2A (0.97) PLAURMEN1KMT2ARAB9ANPC1
SCHEMBL25367120 0.79 KMT2A (0.97) PLAURMEN1KMT2ARAB9ANPC1
SCHEMBL16403339 0.76 PLAUR (0.61) PLAURMEN1KMT2ARAB9ANPC1
SCHEMBL29010071 0.76 PLAUR (0.61) PLAURMEN1KMT2ARAB9ANPC1
SCHEMBL1029154 0.76 PLAUR (0.61) PLAURMEN1KMT2ARAB9ANPC1
SCHEMBL30170557 0.76 PLAUR (0.61) PLAURMEN1KMT2ARAB9ANPC1
SCHEMBL16065887 0.76 PLAUR (0.61) PLAURMEN1KMT2ARAB9ANPC1
SCHEMBL1589916 0.76 PLAUR (0.61) PLAURMEN1KMT2ARAB9ANPC1
SCHEMBL28487096 0.76 PLAUR (0.61) PLAURMEN1KMT2ARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116813593-A 3-aminoquinoxalinone compound and synthesis method thereof 郑州泰基鸿诺医药股份有限公司 2023-09-29 CN claimed
CN-115747838-A Method for synthesizing amino-substituted quinoxalinone compound through electrochemical reaction 南京师范大学 2023-03-07 CN claimed
CN-105001169-A Synthetic method for 3-aminoquinoxaline-2(1H)-ketone compound UNIV HUAQIAO 2015-10-28 CN claimed
EP-1649857-A2 New use of glutamate antagonists for the treatment of cancer Ikonomidou, Hrissanthi (DE) 2006-04-26 EP claimed
US-20050054650-A1 Use of glutamate antagonists for the treatment of cancer IKONOMIDOU HRISSANTHI (DE) 2005-03-10 US claimed
EP-1124553-A1 NEW USE OF GLUTAMATE ANTAGONISTS FOR THE TREATMENT OF CANCER Ikonomidou, Hrissanthi (DE) 2001-08-22 EP claimed
EP-1002535-A1 New use of glutamate antagonists for the treatment of cancer Ikonomidou, Hrissanthi (DE) 2000-05-24 EP claimed
WO-2000024395-A1 NEW USE OF GLUTAMATE ANTAGONISTS FOR THE TREATMENT OF CANCER IKONOMIDOU HRISSANTHI (DE) 2000-05-04 WO claimed
US-5633255-A RESPIRATORY SYSTEM DISORDERS; ACID HYDROLYSIS; ALKYLATION PIERRE FABRE MEDICAMENT (FR) 1997-05-27 US claimed
EP-0663903-B1 1,2-DIHYDRO-2-OXO-3-AMINO QUINOXALINE DERIVATIVES, PREPARATION THEREOF AND APPLICATION IN THERAPY PF MEDICAMENT (FR) 1997-04-23 EP claimed
CN-116813593-A 3-aminoquinoxalinone compound and synthesis method thereof 郑州泰基鸿诺医药股份有限公司 2023-09-29 CN disclosed
CN-116813593-A 3-aminoquinoxalinone compound and synthesis method thereof 郑州泰基鸿诺医药股份有限公司 2023-09-29 CN disclosed
CN-116813593-A 3-aminoquinoxalinone compound and synthesis method thereof 郑州泰基鸿诺医药股份有限公司 2023-09-29 CN disclosed
CN-109160903-B Photocatalytic preparation method of 3-aminoquinoxaline-2 (1H) -ketone compound 曲阜师范大学 2021-07-16 CN disclosed
CN-107973755-B Preparation method of 3-acetamido quinoxalinone derivative 滨州学院 2020-12-29 CN disclosed
WO-1996004288-A1 GLYCINE RECEPTOR ANTAGONIST PHARMACOPHORE STATE OF OREGON, ACTING BY AND THROUGH THE OREGON STATE BOARD OF HIGHER EDUCATION, ACTING FOR AND ON BEHALF OF THE OREGON HEALTH SCIENCES UNIVERSITY AND THE UNIVERSITY OF OREGON, EUGENE OREGON (US) 1996-02-15 WO disclosed
EP-0663903-A1 1,2-DIHYDRO-2-OXO-3-AMINO QUINOXALINE DERIVATIVES, PREPARATION THEREOF AND APPLICATION IN THERAPY. PF MEDICAMENT (FR) 1995-07-26 EP disclosed
WO-1994007870-A1 1,2-DIHYDRO-2-OXO-3-AMINO QUINOXALINE DERIVATIVES, PREPARATION THEREOF AND APPLICATION IN THERAPY PIERRE FABRE MEDICAMENT (FR) 1994-04-14 WO disclosed
EP-0185618-A2 Isoindolines, process for their manufacture and their use CIBA-GEIGY AG (CH) 1986-06-25 EP disclosed
US-3963694-A AZO PIGMENTS, POLYESTERS, CELLULOSE ETHERS AND ESTERS CIBA-GEIGY CORPORATION (US) 1976-06-15 US disclosed