SCHEMBL1898539

SCHEMBL1898539

O=C(O)c1cc(-c2ccc(F)cc2)nc2ccccc12

nearest known ligand 0.80

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 11/20 0.80
KDM4E B2RXH2 1/20 0.79
LMNA P02545 1/20 0.79
SMN1; SMN2 Q16637 1/20 0.79
PDE10A Q9Y233 1/20 0.79
POLB P06746 1/20 0.76
MEN1 O00255 1/20 0.74
NPC1 O15118 1/20 0.74
RAB9A P51151 1/20 0.74
KMT2A Q03164 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29788460 1.00 DHODH (0.80) DHODHKDM4ELMNASMN1; SMN2PDE10A
SCHEMBL29536364 0.89 DHODH (1.00) DHODHKDM4ELMNASMN1; SMN2PDE10A
SCHEMBL2467110 0.89 DHODH (1.00) DHODHKDM4ELMNASMN1; SMN2PDE10A
Cinchophen SCHEMBL25519 0.89 KDM4E (1.00) DHODHKDM4ELMNASMN1; SMN2PDE10A
Cinchophen SCHEMBL7588217 0.89 KDM4E (1.00) DHODHKDM4ELMNASMN1; SMN2PDE10A
Cinchophen SCHEMBL29376617 0.89 KDM4E (1.00) DHODHKDM4ELMNASMN1; SMN2PDE10A
SCHEMBL10867811 0.88 DHODH (0.62) DHODHKDM4ELMNASMN1; SMN2PDE10A
SCHEMBL10436053 0.88 DHODH (0.67) DHODHKDM4ELMNASMN1; SMN2PDE10A
SCHEMBL19537432 0.88 KDM4E (0.74) DHODHKDM4ELMNASMN1; SMN2PDE10A
Cinchophen SCHEMBL4464779 0.87 KDM4E (0.97) DHODHKDM4ELMNASMN1; SMN2PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108250230-B Refining method of diisopropylamine silane 浙江博瑞电子科技有限公司 2020-09-15 CN claimed
EP-4617270-A1 ISOINDOLINONE DERIVATIVE HAVING QUINOLINE AMIDE STRUCTURE, AND USE THEREOF Oncord Bio Inc (KR) 2025-09-17 EP disclosed
WO-2024101764-A1 ISOINDOLINONE DERIVATIVE HAVING QUINOLINE AMIDE STRUCTURE, AND USE THEREOF 주식회사 온코드바이오 2024-05-16 WO disclosed
CN-111574530-B ACC inhibitor and medical application thereof 徐州医科大学 2022-07-26 CN disclosed
CN-108358838-B Novel quinoline-substituted Schiff base derivative with biological activity and synthesis method and application thereof 河南师范大学 2021-05-18 CN disclosed
CN-108250230-B Refining method of diisopropylamine silane 浙江博瑞电子科技有限公司 2020-09-15 CN disclosed
CN-111574530-A ACC inhibitor and medical application thereof 徐州医科大学 2020-08-25 CN disclosed
CN-108250230-A A kind of process for purification of diisopropylamine silane 浙江博瑞电子科技有限公司 2018-07-06 CN disclosed
EP-2325181-B1 STAT3 INHIBITOR CONTAINING QUINOLINECARBOXAMIDE DERIVATIVE AS ACTIVE INGREDIENT GENERAL INCORPORATED ASS PHARMA VALLEY PROJECT SUPPORTING ORGANIZATION (JP) 2017-03-29 EP disclosed
WO-2016202898-A1 GLUCOSE TRANSPORT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-12-22 WO disclosed
WO-2009082346-A1 NEW ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS AND USES IN TREATMENTS OF OBESITY AND DIABETES MELLITUS - 087 ASTRAZENECA AB (SE) 2009-07-02 WO disclosed
WO-2009082346-A1 NEW ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS AND USES IN TREATMENTS OF OBESITY AND DIABETES MELLITUS - 087 ASTRAZENECA AB (SE) 2009-07-02 WO disclosed
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed
US-4711890-A TREATMENT OF ANXIETY STATES OR OF PULMONARY, RENAL, CIRCULATORY OF CARDIOVASCULAR DISORDERS RHONE-POULENC SANTE (FR) 1987-12-08 US disclosed
US-4684652-A TREATING ANXIETY OR CARDIOVASCULAR DISORDERS RHONE-POULENC SANTE (FR) 1987-08-04 US disclosed
EP-0168812-A1 4-Amino-2-phenyl quinolines, methods and intermediates for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1986-01-22 EP disclosed
US-4560692-A ANTICONVULSANTS OR ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1985-12-24 US disclosed
US-4433150-A HYPNBOTICS, ANTICONVULSANTS, TRANQUILIZERS, ANTIDEPRESSANTS, SEDATIVES, ANTIARRHYTHMIA AGENTS PHARMINDUSTRIE (FR) 1984-02-21 US disclosed