SCHEMBL29536364

SCHEMBL29536364

O=C(O)c1cc(-c2ccc(-c3ccccc3)cc2)nc2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 9/20 1.00
KDM4E B2RXH2 2/20 0.93
PDE10A Q9Y233 2/20 0.93
LMNA P02545 1/20 0.93
SMN1; SMN2 Q16637 1/20 0.93
POLB P06746 1/20 0.82
TP53 P04637 1/20 0.75
CYP1A2 P05177 1/20 0.75
CYP2C19 P33261 1/20 0.75
HIF1A Q16665 1/20 0.75
HSD17B10 Q99714 1/20 0.75
AKR1C3 P42330 1/20 0.73
AKR1C2 P52895 1/20 0.73
AKR1C1 Q04828 1/20 0.73
KMT2A Q03164 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2467110 1.00 DHODH (1.00) DHODHKDM4EPDE10ALMNASMN1; SMN2
Cinchophen SCHEMBL29376617 0.97 KDM4E (1.00) DHODHKDM4EPDE10ALMNASMN1; SMN2
Cinchophen SCHEMBL25519 0.97 KDM4E (1.00) DHODHKDM4EPDE10ALMNASMN1; SMN2
Cinchophen SCHEMBL7588217 0.97 KDM4E (1.00) DHODHKDM4EPDE10ALMNASMN1; SMN2
Cinchophen SCHEMBL4805149 0.95 KDM4E (0.97) DHODHKDM4EPDE10ALMNASMN1; SMN2
Cinchophen SCHEMBL10757475 0.95 KDM4E (0.97) DHODHKDM4EPDE10ALMNASMN1; SMN2
Cinchophen SCHEMBL4464779 0.95 KDM4E (0.97) DHODHKDM4EPDE10ALMNASMN1; SMN2
Cinchophen SCHEMBL27543969 0.93 KDM4E (0.93) DHODHKDM4EPDE10ALMNASMN1; SMN2
SCHEMBL3237037 0.90 POLB (1.00) DHODHKDM4EPDE10ALMNASMN1; SMN2
SCHEMBL8689228 0.90 DHODH (0.82) DHODHKDM4EPDE10ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117050110-A GPX4 and DHODH double-inhibition small molecule prodrug compound based on mitochondrial targeting and preparation method and application thereof 厦门大学 2023-11-14 CN claimed
CN-117327011-A Quinoline PCSK9 inhibitor and preparation method and application thereof 山东省分析测试中心 2024-01-02 CN disclosed
CN-117050110-A GPX4 and DHODH double-inhibition small molecule prodrug compound based on mitochondrial targeting and preparation method and application thereof 厦门大学 2023-11-14 CN disclosed
EP-3976594-A1 A THERAPEUTIC APPROACH FOR TREATING NON-INFECTIOUS OCULAR IMMUNOINFLAMMATORY DISORDERS The Schepens Eye Research Institute, Inc. (US) 2022-04-06 EP disclosed