SCHEMBL19001693

SCHEMBL19001693

Clc1ccc2c(c1)C1(c3ccccc3-c3c(-c4ccccc4)cccc31)c1cccc(Br)c1-2

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 12/20 0.42
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
AKR1A1 P14550 1/20 0.36
AKR1B1 P15121 1/20 0.36
SLC6A3 Q01959 1/20 0.34
PTGES O14684 1/20 0.32
CYP2A6 P11509 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31497074 0.90 PDK2 (0.44) PDK2AKR1A1AKR1B1SLC6A3CYP2A6
SCHEMBL20680539 0.90 PDK2 (0.44) PDK2AKR1A1AKR1B1SLC6A3CYP2A6
SCHEMBL19001688 0.90 PDK2 (0.47) PDK2ALDH1A1AKR1A1AKR1B1PTGES
SCHEMBL28886028 0.90 PDK2 (0.44) PDK2AKR1A1AKR1B1SLC6A3CYP2A6
SCHEMBL19001700 0.90 PDK2 (0.39) PDK2ALDH1A1MAPK1AKR1A1AKR1B1
SCHEMBL19001692 0.90 PDK2 (0.44) PDK2AKR1A1AKR1B1
SCHEMBL20687347 0.90 PDK2 (0.40) PDK2ALDH1A1MAPK1AKR1A1AKR1B1
SCHEMBL20687306 0.89 PDK2 (0.44) PDK2AKR1A1AKR1B1SLC6A3CYP2A6
SCHEMBL20687322 0.88 PDK2 (0.43) PDK2AKR1A1AKR1B1SLC6A3
SCHEMBL19001863 0.87 PDK2 (0.49) PDK2ALDH1A1MAPK1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3390365-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2021-04-14 EP disclosed
WO-2017102063-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2017-06-22 WO disclosed