SCHEMBL19004902

SCHEMBL19004902

Nc1ccc(-c2cnn(CC3CC3(F)F)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.40
PIK3CA P42336 2/20 0.40
PIK3CB P42338 2/20 0.40
PI4KA P42356 2/20 0.40
PIK3CG P48736 2/20 0.40
PI4KB Q9UBF8 2/20 0.40
BRD4 O60885 1/20 0.37
CREBBP Q92793 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
KDM1A O60341 1/20 0.35
KCNH2 Q12809 4/20 0.35
TBK1 Q9UHD2 3/20 0.35
FEN1 P39748 1/20 0.33
METAP2 P50579 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
LRRK2 Q5S007 1/20 0.33
ALOX5AP P20292 1/20 0.32
TYRO3 Q06418 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18985752 0.85 PIK3CD (0.43) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL19005256 0.79 PIK3CD (0.39) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL18985778 0.78 TBK1 (0.38) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL18985609 0.77 MAPT (0.48) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL18985433 0.77 TBK1 (0.39) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL19668078 0.76 FFAR1 (0.38) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL19668107 0.75 LRRK2 (0.34) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL12090082 0.73 TBK1 (0.33) TBK1
SCHEMBL18985666 0.72 PIK3CD (0.44) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL6920523 0.72 ALPI (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102091-A1 HETEROARYLBENZIMIDAZOLE COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-22 WO disclosed