SCHEMBL19005672

SCHEMBL19005672

O=c1nccc2n1CCNC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 10/20 0.40
HTR2A P28223 8/20 0.40
HRH3 Q9Y5N1 1/20 0.33
PLD1 Q13393 2/20 0.33
ADRB2 P07550 2/20 0.32
NCF1 P14598 2/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 1/20 0.32
KDM5C P41229 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
MEN1 O00255 1/20 0.31
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALOX15 P16050 1/20 0.31
MAPK1 P28482 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14659998 0.72 HSD17B10 (0.37) KDM4EALDH1A1CYP1A2CYP3A4MAPT
SCHEMBL27957909 0.71 MCHR1 (0.35) HTR2CHTR2AHRH3PLD1ADRB2
SCHEMBL12214112 0.70 HTR2C (0.46) HTR2CHTR2AKDM4EMEN1TP53
SCHEMBL14975241 0.70 MEN1 (0.35) KDM4EALDH1A1MEN1MAPTMAPK1
SCHEMBL31372266 0.68 PIK3CA (0.33) ALDH1A1
SCHEMBL928949 0.67 HTR7 (0.47) HTR2CHTR2APLD1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL25413336 0.67 HTR2C (0.40) HTR2CHTR2AKDM4EMEN1TP53
SCHEMBL26914967 0.66 HTR2C (0.42) HTR2CHTR2AKDM4EALDH1A1MEN1
SCHEMBL929336 0.66 HTR2A (0.36) HTR2CHTR2APLD1ADRB2NCF1
SCHEMBL928542 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017101796-A1 PHTHALAZINONE DERIVATIVE, AND PREPARATION METHOD AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed