SCHEMBL19005706

SCHEMBL19005706

Cn1cc(-c2nnc3n2CCN(C(=O)OC(C)(C)C)C3)cn1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RET P07949 8/20 0.46
TTK P33981 1/20 0.46
GPR119 Q8TDV5 1/20 0.46
PDK2 Q15119 1/20 0.44
LRRK2 Q5S007 1/20 0.44
PARP1 P09874 1/20 0.43
USP30 Q70CQ3 2/20 0.43
NR1H2 P55055 1/20 0.42
PIK3CD O00329 1/20 0.41
MET P08581 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28886725 0.83 PDK2 (0.47) RETTTKGPR119PDK2LRRK2
SCHEMBL12461826 0.82 RET (0.55) RETTTK
SCHEMBL20157515 0.82 PDK2 (0.64) PDK2NR1H2
SCHEMBL19005627 0.81 P2RX7 (0.58) RETTTKPDK2PARP1NR1H2
SCHEMBL10095021 0.79 NR1H2 (0.47) PDK2NR1H2
SCHEMBL16027918 0.77 P2RX7 (0.59) GPR119
SCHEMBL30552179 0.76 P2RX7 (0.56)
SCHEMBL26113816 0.76 P2RX7 (0.56)
SCHEMBL109572 0.75 TACR3 (0.41) TTKPDK2NR1H2
SCHEMBL30980030 0.75 P2RX7 (0.56) GPR119PDK2PARP1NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017101796-A1 PHTHALAZINONE DERIVATIVE, AND PREPARATION METHOD AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed