SCHEMBL19006591

SCHEMBL19006591

COC(=O)CC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(Cl)cc1C(=O)c1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR9 P51686 2/20 0.45
GRM5 P41594 2/20 0.39
HDAC4 P56524 4/20 0.39
HDAC1 Q13547 4/20 0.39
CTSL P07711 1/20 0.39
HDAC3 O15379 2/20 0.38
HDAC7 Q8WUI4 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC10 Q969S8 2/20 0.38
HDAC11 Q96DB2 2/20 0.38
HDAC8 Q9BY41 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
HDAC9 Q9UKV0 2/20 0.38
HDAC5 Q9UQL6 2/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20473233 1.00 CCR9 (0.45) CCR9GRM5HDAC4HDAC1CTSL
SCHEMBL20473216 0.92 CCR9 (0.44) CCR9GRM5HDAC4HDAC1CTSL
SCHEMBL17244394 0.90 AAK1 (0.45) HDAC4HDAC1HDAC3HDAC7HDAC2
SCHEMBL20680744 0.90 AAK1 (0.45) HDAC4HDAC1HDAC3HDAC7HDAC2
SCHEMBL29368604 0.90 AAK1 (0.45) HDAC4HDAC1HDAC3HDAC7HDAC2
SCHEMBL22853706 0.87 HDAC1 (0.41) HDAC4HDAC1CTSLHDAC3HDAC7
SCHEMBL20473276 0.87 SMN1; SMN2 (0.47) ALDH1A1SMN1; SMN2MAPTGAA
SCHEMBL19006724 0.87 SMN1; SMN2 (0.47) ALDH1A1SMN1; SMN2MAPTGAA
SCHEMBL22591862 0.85 HDAC4 (0.40) HDAC4HDAC1HDAC3HDAC7HDAC2
SCHEMBL20473299 0.85 CTSS (0.41) HDAC4HDAC1CTSLHDAC3HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017101808-A1 SHORT-ACTING BENZODIAZEPINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed