SCHEMBL19006745

SCHEMBL19006745

COC(=O)CC[C@@H]1N=C(c2ccccn2)c2cc(Br)ccc2N=C1O[PH](=O)N1CCOCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 2/20 0.32
TP53 P04637 2/20 0.32
RAB9A P51151 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
NPY1R P25929 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
ALOX15 P16050 1/20 0.32
KMT2A Q03164 1/20 0.32
BRD4 O60885 1/20 0.31
BACE1 P56817 1/20 0.31
SCN5A Q14524 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19006599 0.91
SCHEMBL13862620 0.88
SCHEMBL17244387 0.86 LMNA (0.34) LMNANPSR1TDP1L3MBTL1NPC1
SCHEMBL17166207 0.85 LMNA (0.34) LMNANPSR1TDP1L3MBTL1NPC1
SCHEMBL20473341 0.85 LMNA (0.34) LMNANPSR1TDP1L3MBTL1NPC1
SCHEMBL14329002 0.83 LMNA (0.33) LMNANPSR1TDP1L3MBTL1NPC1
SCHEMBL20907118 0.81 NPY1R (0.35) NPC1TP53RAB9ASMN1; SMN2NPY1R
SCHEMBL21454863 0.79 KDM4E (0.36) NPC1TP53RAB9ASMN1; SMN2KDM4E
SCHEMBL20906913 0.79 NPY1R (0.35) NPC1TP53RAB9ASMN1; SMN2NPY1R
SCHEMBL13862621 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017101808-A1 SHORT-ACTING BENZODIAZEPINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed