SCHEMBL19006944

SCHEMBL19006944

COc1cc2c(Nc3ccc(Br)cc3C)ncnc2cc1OCC1CCOCC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.72
EPHA2 P29317 9/20 0.72
EPHB4 P54760 6/20 0.72
EGFR P00533 9/20 0.65
FGFR1 P11362 6/20 0.65
FLT1 P17948 6/20 0.65
FLT4 P35916 6/20 0.65
RET P07949 3/20 0.65
PDGFRB P09619 2/20 0.65
TEK Q02763 2/20 0.65
ERBB2 P04626 2/20 0.65
KIF5B P33176 2/20 0.65
BMPR1B O00238 1/20 0.65
PLK4 O00444 1/20 0.65
CIT O14578 1/20 0.65
GAK O14976 1/20 0.65
EPHB6 O15197 1/20 0.65
RIPK2 O43353 1/20 0.65
ROCK2 O75116 1/20 0.65
STK10 O94804 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17520370 0.90 KDR (0.79) KDREPHA2EPHB4EGFRFGFR1
SCHEMBL18211400 0.88 EGFR (0.82) KDREPHA2EPHB4EGFRFGFR1
SCHEMBL22592730 0.87 KDR (0.75) KDREPHA2EPHB4EGFRFGFR1
SCHEMBL19220787 0.85 EGFR (0.81) KDREPHA2EPHB4EGFRFGFR1
SCHEMBL1791359 0.84 EPHA2 (1.00) KDREPHA2EPHB4EGFRERBB2
SCHEMBL19154592 0.80 EGFR (0.84) KDREPHA2EPHB4EGFRFGFR1
SCHEMBL1612820 0.79 KDR (0.84) KDREPHA2EPHB4EGFRFGFR1
SCHEMBL31319937 0.79 KDR (0.84) KDREPHA2EPHB4EGFRFGFR1
Vandetanib SCHEMBL9044 0.79 EGFR (1.00) KDREPHA2EPHB4EGFRFGFR1
Vandetanib SCHEMBL29352879 0.79 EGFR (1.00) KDREPHA2EPHB4EGFRFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3181554-A1 QUINAZOLINE DERIVATIVE CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang) Co., Ltd. (CN) 2017-06-21 EP disclosed