SCHEMBL19006973

SCHEMBL19006973

COc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cc1CCCCCCN(C)C

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.76
KDR P35968 2/20 0.67
FBP1 P09467 2/20 0.67
AURKA O14965 1/20 0.67
ERBB2 P04626 1/20 0.67
INSR P06213 1/20 0.67
PDGFRB P09619 1/20 0.67
FLT4 P35916 1/20 0.67
CLK1 P49759 1/20 0.67
EPHB4 P54760 1/20 0.67
TEK Q02763 1/20 0.67
AURKB Q96GD4 1/20 0.67
HDAC3 O15379 1/20 0.67
HDAC4 P56524 1/20 0.67
HDAC1 Q13547 1/20 0.67
HDAC7 Q8WUI4 1/20 0.67
HDAC2 Q92769 1/20 0.67
HDAC10 Q969S8 1/20 0.67
HDAC11 Q96DB2 1/20 0.67
HDAC8 Q9BY41 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17520361 0.87 EGFR (0.94) EGFRKDRFBP1AURKAERBB2
SCHEMBL19006650 0.87 HDAC3 (0.74) EGFRKDRFBP1AURKAERBB2
SCHEMBL17520337 0.86 EGFR (1.00) EGFRKDRFBP1AURKAERBB2
SCHEMBL2102985 0.86 EGFR (1.00) EGFRKDRFBP1AURKAERBB2
SCHEMBL11113 0.83 EGFR (1.00) EGFRKDRFBP1AURKAERBB2
SCHEMBL10118734 0.81 HDAC3 (0.84) EGFRKDRFBP1AURKAERBB2
SCHEMBL30505605 0.81 EGFR (1.00) EGFRKDRFBP1AURKAERBB2
SCHEMBL2099106 0.81 EGFR (1.00) EGFRKDRFBP1AURKAERBB2
SCHEMBL19006953 0.81 KDR (0.67) EGFRKDRERBB2PDGFRBFLT4
SCHEMBL8210222 0.81 HDAC3 (0.98) EGFRKDRERBB2HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3181554-A1 QUINAZOLINE DERIVATIVE CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang) Co., Ltd. (CN) 2017-06-21 EP disclosed