SCHEMBL1900974

SCHEMBL1900974

O=C(O)NC1(c2ccc(-c3oc4nc(N5CCOCC5)ncc4c3-c3ccccc3)cc2)CCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
HSD17B10 Q99714 6/20 0.41
HPGD P15428 4/20 0.41
TSHR P16473 3/20 0.41
PTPN11 Q06124 1/20 0.39
OPRL1 P41146 2/20 0.39
DGAT1 O75907 1/20 0.38
OPRM1 P35372 1/20 0.37
MTOR P42345 3/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CG P48736 1/20 0.37
KDM4E B2RXH2 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CASP1 P29466 2/20 0.36
CASP7 P55210 2/20 0.36
TNK2 Q07912 2/20 0.36
GLA P06280 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1900566 0.91 LCK (0.37) ALDH1A1HSD17B10HPGDOPRL1OPRM1
SCHEMBL1902658 0.84 ALDH1A1 (0.41) ALDH1A1HSD17B10HPGDTSHROPRL1
SCHEMBL1904461 0.84 AKT1 (0.47) ALDH1A1HSD17B10HPGDTSHRMTOR
SCHEMBL14118620 0.83 CKS1B (0.47) OPRM1
SCHEMBL1905448 0.82 TACR3 (0.38) CYP3A4TNK2MAPK1TACR3EGFR
SCHEMBL1904913 0.82 ALDH1A1 (0.41) ALDH1A1HSD17B10HPGDTSHRMTOR
SCHEMBL14118682 0.81 AKT1 (0.41) ALDH1A1HSD17B10HPGDPTPN11OPRL1
SCHEMBL1908151 0.80 TACR3 (0.37) TSHRKDM4EMAPTTACR3POLB
SCHEMBL1902848 0.80 TACR3 (0.37) TNK2MAPK1MAPTTACR3
SCHEMBL14119122 0.79 CKS1B (0.48) OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120309739-A1 AKT / PKB INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2012-12-06 US disclosed
EP-2496566-A1 AKT / PKB INHIBITORS Almac Discovery Limited (GB) 2012-09-12 EP disclosed
WO-2011055115-A1 AKT / PKB INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2011-05-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120309739-A1 AKT / PKB INHIBITORS AKT1, AKT2, AKT3 ALDH1A1 4803/4885HSD17B10 2043/4885HPGD 3200/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.