SCHEMBL1901129

SCHEMBL1901129

O=Cc1ccccc1OC1CCN(C(=O)O)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NPY1R P25929 1/20 0.41
NPY2R P49146 1/20 0.41
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 1/20 0.40
RAD52 P43351 1/20 0.40
HMOX1 P09601 1/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
RBP4 P02753 2/20 0.39
SCN1A P35498 1/20 0.39
SCN2A Q99250 1/20 0.39
SCN3A Q9NY46 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1902995 0.92 HRH1 (0.45) HRH1PTGDR2SMN1; SMN2KDM4ENPY1R
SCHEMBL18043823 0.89 PTGDR2 (0.46) HRH1PTGDR2SMN1; SMN2NPC1MAPT
SCHEMBL1894331 0.83 USP30 (0.50)
SCHEMBL8419333 0.82 GAA (0.57) SMN1; SMN2KDM4ENPY2RNPC1RAB9A
SCHEMBL24590454 0.81 NAMPT (0.47) MAPTKMT2AMEN1ALDH1A1SCD
SCHEMBL24590680 0.81 TEAD3 (0.47) HRH1KMT2ARBP4SCD
SCHEMBL28278842 0.81 EPHX2 (0.57) HRH1SMN1; SMN2KDM4ENPY1RNPY2R
SCHEMBL5114227 0.81 HPGD (0.47) SMN1; SMN2KDM4ENPY1RNPY2RKMT2A
SCHEMBL28086838 0.80 PTGDR2 (0.37) PTGDR2SMN1; SMN2NPC1MAPTRAB9A
SCHEMBL24590535 0.80 NAMPT (0.49) SMN1; SMN2KMT2AMEN1SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2315763-A1 BENZIMIDAZOLES AND RELATED ANALOGS AS SIRTUIN MODULATORS Sirtris Pharmaceuticals, Inc. (US) 2011-05-04 EP disclosed
WO-2010003048-A1 BENZIMIDAZOLES AND RELATED ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2010-01-07 WO disclosed