SCHEMBL19019607

SCHEMBL19019607

Cc1ccc(-c2ccc(-c3ccc(-c4cc(C)c(F)c(F)c4)c(F)c3)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 4/20 0.40
PDE3A Q14432 4/20 0.40
RPS6KA3 P51812 3/20 0.39
PDK2 Q15119 1/20 0.39
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
PTGS2 P35354 6/20 0.37
PTGS1 P23219 2/20 0.36
DAPK3 O43293 1/20 0.36
NTRK1 P04629 1/20 0.36
PIM1 P11309 1/20 0.36
FLT3 P36888 1/20 0.36
GSK3B P49841 1/20 0.36
ROCK1 Q13464 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
AKR1B10 O60218 1/20 0.35
AKR1C4 P17516 1/20 0.35
AKR1C1 Q04828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18973377 1.00 PDE3B (0.40) PDE3BPDE3ARPS6KA3PDK2AKR1C3
SCHEMBL20976650 0.93 RPS6KA3 (0.39) PDE3BPDE3ARPS6KA3PDK2AKR1C3
SCHEMBL2741547 0.91 PDE3B (0.42) PDE3BPDE3ARPS6KA3PDK2AKR1C3
SCHEMBL2741562 0.91 PDE3B (0.42) PDE3BPDE3ARPS6KA3PDK2AKR1C3
SCHEMBL13295485 0.89 PDE3B (0.41) PDE3BPDE3ARPS6KA3PDK2AKR1C3
SCHEMBL17471815 0.88 PTGS2 (0.36) PDE3BPDE3ARPS6KA3PDK2AKR1C3
SCHEMBL13480360 0.87 PDE3B (0.40) PDE3BPDE3ARPS6KA3PDK2AKR1C3
SCHEMBL18973378 0.86 PDE3B (0.40) PDE3BPDE3ARPS6KA3PDK2AKR1C3
SCHEMBL170435 0.85 PDE3B (0.49) PDE3BPDE3ARPS6KA3PDK2AKR1C3
SCHEMBL21373998 0.84 PTGS2 (0.45) PDE3BPDE3ARPS6KA3PDK2AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102053-A2 CINNAMIC ACID DERIVATIVES MERCK PATENT GMBH (DE) 2017-06-22 WO disclosed