SCHEMBL190241

SCHEMBL190241

O=Cc1cc2c(N3CCOCC3)nc(Cl)nc2s1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.48
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
MAPK1 P28482 2/20 0.44
HSD17B10 Q99714 2/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
ALDH3A1 P30838 1/20 0.40
ALDH1A3 P47895 1/20 0.40
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
KMT2A Q03164 1/20 0.38
MAT2A P31153 1/20 0.38
HRH3 Q9Y5N1 3/20 0.38
MAPT P10636 2/20 0.38
PIK3CA P42336 3/20 0.37
PIK3CB P42338 3/20 0.37
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13059942 0.85 KDM4E (0.61) SMN1; SMN2KDM4EALDH1A1HPGDMAPK1
SCHEMBL4446531 0.85 SMN1; SMN2 (0.51) SMN1; SMN2KDM4EALDH1A1HPGDMAPK1
SCHEMBL4441865 0.82 SMN1; SMN2 (0.49) SMN1; SMN2KDM4EALDH1A1HPGDMAPK1
SCHEMBL8199168 0.82 SMN1; SMN2 (0.49) SMN1; SMN2KDM4EALDH1A1HPGDMAPK1
SCHEMBL1856986 0.81 PIK3CA (0.52) SMN1; SMN2KDM4EALDH1A1HPGDMAPK1
SCHEMBL4434053 0.80 PIK3CA (0.50) SMN1; SMN2KDM4EALDH1A1HPGDMAPK1
SCHEMBL1860340 0.80 SMN1; SMN2 (0.44) SMN1; SMN2KDM4EALDH1A1HPGDMAPK1
SCHEMBL189813 0.78 PIK3CA (0.49) SMN1; SMN2ALDH3A1ALDH1A3PIK3CAPIK3CB
SCHEMBL4068550 0.78 SMN1; SMN2 (0.45) SMN1; SMN2KDM4EALDH1A1HPGDMAPK1
SCHEMBL1859364 0.78 SMN1; SMN2 (0.48) SMN1; SMN2KDM4EALDH1A1HPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 130 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101909631-B Process for making thienopyrimidine compounds GENENTECH INC 2012-09-12 CN claimed
US-20100292468-A1 PROCESS FOR MAKING THIENOPYRIMIDINE COMPOUNDS GENETECH, INC 2010-11-18 US claimed
EP-2214675-A1 PROCESS FOR MAKING THIENOPYRIMIDINE COMPOUNDS Genentech, Inc. (US) 2010-08-11 EP claimed
WO-2009055730-A1 PROCESS FOR MAKING THIENOPYRIMIDINE COMPOUNDS GENENTECH, INC. (US) 2009-04-30 WO claimed
US-11603372-B2 Compounds and therapeutic uses thereof VIOGEN BIOSCIENCES, LLC (US) 2023-03-14 US disclosed
US-20210122752-A1 COMPOUNDS AND THERAPEUTIC USES THEREOF VIOGEN BIOSCIENCES, LLC 2021-04-29 US disclosed
US-20210122752-A1 COMPOUNDS AND THERAPEUTIC USES THEREOF VIOGEN BIOSCIENCES, LLC 2021-04-29 US disclosed
WO-2019113523-A1 COMPOUNDS AND THERAPEUTIC USES THEREOF BAJJI ASHOK (US) 2019-06-13 WO disclosed
WO-2019113523-A1 COMPOUNDS AND THERAPEUTIC USES THEREOF BAJJI ASHOK (US) 2019-06-13 WO disclosed
US-9943519-B2 Pharmaceutical compounds GENENTECH, INC. (US) 2018-04-17 US disclosed
US-9943519-B2 Pharmaceutical compounds GENENTECH, INC. (US) 2018-04-17 US disclosed
US-9943519-B2 Pharmaceutical compounds GENENTECH, INC. (US) 2018-04-17 US disclosed
US-20080039459-A1 Phosphoinositide 3-kinase inhibitor compounds and methods of use PLRAMED LIMITED (GB) 2008-02-14 US disclosed
US-20080039459-A1 Phosphoinositide 3-kinase inhibitor compounds and methods of use PLRAMED LIMITED (GB) 2008-02-14 US disclosed
US-20080039459-A1 Phosphoinositide 3-kinase inhibitor compounds and methods of use PLRAMED LIMITED (GB) 2008-02-14 US disclosed
WO-2007127183-A1 PHOSPHOINOSITIDE 3-KINASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GENENTECH, INC. (US) 2007-11-08 WO disclosed
WO-2007127183-A1 PHOSPHOINOSITIDE 3-KINASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GENENTECH, INC. (US) 2007-11-08 WO disclosed
WO-2007127175-A2 PHARMACEUTICAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2007-11-08 WO disclosed
WO-2007127175-A2 PHARMACEUTICAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2007-11-08 WO disclosed
WO-2007122410-A1 PYRIMIDINE DERIVATIVES AS PI3K INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-11-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100292468-A1 PROCESS FOR MAKING THIENOPYRIMIDINE COMPOUNDS PIK3CA, PIK3CD, PIK3CB SMN1; SMN2 3575/4885KDM4E 1752/4885ALDH1A1 1766/4885
US-20080039459-A1 Phosphoinositide 3-kinase inhibitor compounds and methods of use PIK3CA, PI4KB, PI4KA SMN1; SMN2 1774/4885KDM4E 3626/4885ALDH1A1 2960/4885
US-11603372-B2 Compounds and therapeutic uses thereof IL15, IL17A, IL2 SMN1; SMN2 1341/4885KDM4E 3881/4885ALDH1A1 1513/4885
US-20210122752-A1 COMPOUNDS AND THERAPEUTIC USES THEREOF IL15, IL17A, IL2 SMN1; SMN2 1341/4885KDM4E 3881/4885ALDH1A1 1513/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.