SCHEMBL19028362

SCHEMBL19028362

C[C@@H](O)c1ccc(F)c(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT2B7 P16662 1/20 0.44
PARP1 P09874 2/20 0.40
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
ADRB1 P08588 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRB3 P13945 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
ADRB2 P07550 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
NOX1 Q9Y5S8 1/20 0.34
EPAS1 Q99814 1/20 0.34
RECQL P46063 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850794 1.00 UGT2B7 (0.44) UGT2B7PARP1KMT2AMEN1ADRB1
SCHEMBL8220975 1.00 UGT2B7 (0.44) UGT2B7PARP1KMT2AMEN1ADRB1
SCHEMBL29903264 0.83 UGT2B7 (0.44) UGT2B7KMT2AMEN1ADRA2BADRB2
SCHEMBL14966853 0.83 UGT2B7 (0.44) UGT2B7KMT2AMEN1ADRA2BADRB2
SCHEMBL3709776 0.83 PARP1 (0.36) PARP1ADRB1ADRA2AADRB3ADRA2B
SCHEMBL31550151 0.83 PARP1 (0.42) PARP1LMNAHIF1A
SCHEMBL8243510 0.83 PARP1 (0.42) PARP1LMNAHIF1A
SCHEMBL4444491 0.81 PARP1 (0.41) PARP1ADRB1ADRA2AADRB3ADRA2B
SCHEMBL248016 0.80 PARP1 (0.40) PARP1ADRB2CYP1A2CYP2D6CYP2C9
SCHEMBL30726196 0.80 PARP1 (0.40) PARP1ADRB2CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017108204-A1 NOVEL SUBSTITUTED SPIRO-[INDOLINE HETEROCYCLOALKANE] COMPOUNDS AS PHOSPHODIESTERASE INHIBITORS Grünenthal GmbH (DE) 2017-06-29 WO disclosed