SCHEMBL19059261

SCHEMBL19059261

CCOc1ccc(CC(=O)N2CCC2)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.52
GPR119 Q8TDV5 6/20 0.52
ALDH1A1 P00352 1/20 0.50
HSD17B10 Q99714 1/20 0.50
HPGD P15428 2/20 0.48
KDM4E B2RXH2 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
FKBP1A P62942 1/20 0.45
CPS1 P31327 3/20 0.44
RAB9A P51151 1/20 0.44
HTR2A P28223 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24437726 0.97 HPGD (0.51) KCNH2GPR119ALDH1A1HSD17B10HPGD
SCHEMBL19059471 0.82 KCNH2 (0.45) KCNH2GPR119L3MBTL1FKBP1ACPS1
SCHEMBL13195634 0.81 KCNH2 (0.42) KCNH2GPR119CPS1HTR2A
SCHEMBL13195630 0.79 DPP4 (0.52) KCNH2GPR119ALDH1A1HSD17B10HPGD
SCHEMBL19058661 0.79 NAMPT (0.40) KCNH2GPR119CPS1HTR2A
SCHEMBL19059444 0.77 SMN1; SMN2 (0.62) ALDH1A1HSD17B10HPGDKDM4EL3MBTL1
SCHEMBL14968299 0.77 KMT2A (0.48) KCNH2GPR119RAB9A
SCHEMBL31481058 0.77 PARP10 (0.47) ALDH1A1KDM4ECPS1HTR2A
SCHEMBL19059479 0.77 KMT2A (0.38) KCNH2GPR119ALDH1A1CPS1HTR2A
SCHEMBL13195638 0.77 KCNH2 (0.39) KCNH2GPR119CPS1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2693882-B1 SUBSTITUTED CYCLOPROPYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT MERCK SHARP & DOHME (US) 2017-06-28 EP disclosed