SCHEMBL19059356

SCHEMBL19059356

CC(C)(C)COCn1ccc2c(-c3cn[nH]c3)ncnc21

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.40
PRMT5 O14744 1/20 0.34
SCN9A Q15858 1/20 0.33
CHUK O15111 6/20 0.31
TPH1 P17752 1/20 0.30
PIK3CG P48736 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99142 0.83 SIGMAR1 (0.40) SIGMAR1PRMT5SCN9ATPH1
SCHEMBL31089960 0.83 SIGMAR1 (0.40) SIGMAR1PRMT5SCN9ATPH1
SCHEMBL21201777 0.82 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ATPH1
SCHEMBL17539275 0.82 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ATPH1
SCHEMBL19928567 0.82 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ATPH1PIK3CG
SCHEMBL13286173 0.82 SIGMAR1 (0.46) SIGMAR1PRMT5SCN9ACHUKTPH1
SCHEMBL17387449 0.81 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ATPH1
SCHEMBL871452 0.81 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ACHUKTPH1
SCHEMBL30749810 0.81 SIGMAR1 (0.39) SIGMAR1PRMT5SCN9ACHUKTPH1
SCHEMBL19790150 0.81 SIGMAR1 (0.38) SIGMAR1PRMT5SCN9ACHUKTPH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017109524-A1 METHOD AND INTERMEDIATE FOR THE PRODUCTION OF BARICITINIB EGIS GYÓGYSZERGYÁR ZRT. (HU) 2017-06-29 WO disclosed