SCHEMBL19062148

SCHEMBL19062148

C/C=C/N(C)c1nc(-c2ccnc3[nH]ccc23)cs1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 5/20 0.46
CIT O14578 1/20 0.45
ROCK1 Q13464 5/20 0.44
PRKCI P41743 2/20 0.44
CCNK O75909 2/20 0.40
CDK12 Q9NYV4 2/20 0.40
JAK2 O60674 2/20 0.40
PRKACA P17612 2/20 0.40
JAK3 P52333 2/20 0.40
PRKCQ Q04759 2/20 0.40
IKBKB O14920 2/20 0.40
AURKB Q96GD4 2/20 0.40
CHUK O15111 1/20 0.40
DAPK3 O43293 1/20 0.40
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
PAK4 O96013 1/20 0.40
CSF1R P07333 1/20 0.40
RET P07949 1/20 0.40
IGF1R P08069 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18602197 0.85 NUDT1 (0.52) NUDT1CITROCK1PRKCICCNK
SCHEMBL99688 0.79 NUDT1 (0.49) NUDT1CITROCK1PRKCICCNK
SCHEMBL29540606 0.79 ROCK1 (0.52) NUDT1CITROCK1PRKCICCNK
SCHEMBL99400 0.79 ROCK1 (0.52) NUDT1CITROCK1PRKCICCNK
SCHEMBL12257978 0.76 NUDT1 (0.56) NUDT1CITROCK1PRKCICCNK
Trifluoroacetic Acid SCHEMBL29540745 0.71 ROCK1 (0.48) NUDT1CITROCK1PRKCICCNK
Trifluoroacetic Acid SCHEMBL5145042 0.71 ROCK1 (0.48) NUDT1CITROCK1PRKCICCNK
SCHEMBL98272 0.69 ROCK1 (0.62) NUDT1CITROCK1PRKCICCNK
SCHEMBL14494761 0.69 NUDT1 (0.64) NUDT1CITROCK1PRKCICCNK
SCHEMBL29541527 0.68 ROCK1 (0.63) NUDT1CITROCK1PRKCICCNK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3838903-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVE AS JANUS KINASE INHIBITOR Incyte Holdings Corporation (US) 2021-06-23 EP disclosed
EP-3466953-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVE AS JANUS KINASE INHIBITOR Incyte Holdings Corporation (US) 2019-04-10 EP disclosed
EP-3184526-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS JANUS KINASE INHIBITOR Incyte Holdings Corporation (US) 2017-06-28 EP disclosed