SCHEMBL19062191

SCHEMBL19062191

C#CCC(c1cccc(C#N)c1)n1cc(-c2ncnc3c2ccn3CC)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 1/20 0.40
JAK2 O60674 7/20 0.36
JAK1 P23458 6/20 0.36
TP53 P04637 1/20 0.33
ABL1 P00519 3/20 0.33
DAPK3 O43293 2/20 0.33
PAK4 O96013 2/20 0.33
RET P07949 2/20 0.33
LTK P29376 2/20 0.33
CSNK1A1 P48729 2/20 0.33
CLK2 P49760 2/20 0.33
JAK3 P52333 2/20 0.33
TNK2 Q07912 2/20 0.33
ROCK1 Q13464 2/20 0.33
DYRK1A Q13627 2/20 0.33
IKBKE Q14164 2/20 0.33
NTRK3 Q16288 2/20 0.33
NTRK2 Q16620 2/20 0.33
LRRK2 Q5S007 2/20 0.33
TAOK1 Q7L7X3 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL100894 0.87 CREBBP (0.37) CREBBPJAK2JAK1
SCHEMBL18638785 0.86 CREBBP (0.39) CREBBPJAK2JAK1RPS6KB1
SCHEMBL102811 0.80 JAK2 (0.53) JAK2JAK1ABL1DAPK3PAK4
SCHEMBL13678307 0.76 JAK2 (0.54) CREBBPJAK2JAK1ABL1DAPK3
Trifluoroacetic Acid SCHEMBL29540688 0.75 TYRO3 (0.50) JAK2JAK1ABL1DAPK3PAK4
Trifluoroacetic Acid SCHEMBL100597 0.75 TYRO3 (0.50) JAK2JAK1ABL1DAPK3PAK4
SCHEMBL101788 0.75 CREBBP (0.37) CREBBPJAK2JAK1LRRK2TYRO3
SCHEMBL15267801 0.74 JAK2 (0.56) JAK2JAK1ABL1DAPK3PAK4
SCHEMBL19075430 0.74 JAK2 (0.44) JAK2JAK1ABL1DAPK3PAK4
SCHEMBL2144942 0.73 JAK2 (0.59) JAK2JAK1ABL1DAPK3PAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3184526-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS JANUS KINASE INHIBITOR Incyte Holdings Corporation (US) 2017-06-28 EP disclosed