SCHEMBL19063000

SCHEMBL19063000

NC(CF)Cc1ccc(-c2cnccn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.43
CYP19A1 P11511 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
BRS3 P32247 1/20 0.41
PIM1 P11309 1/20 0.37
PIM2 Q9P1W9 1/20 0.37
AKT1 P31749 5/20 0.37
CDK2 P24941 5/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PI4KA P42356 1/20 0.37
PIK3CG P48736 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
MET P08581 1/20 0.36
WNT3A P56704 2/20 0.36
MAPT P10636 1/20 0.36
HDAC4 P56524 1/20 0.36
CA12 O43570 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31140237 0.78 CYP2D6 (0.51) CYP2D6CYP19A1CYP2C9CYP2C19BRS3
SCHEMBL10130785 0.78 CYP2D6 (0.51) CYP2D6CYP19A1CYP2C9CYP2C19BRS3
SCHEMBL4750423 0.77 CYP2A6 (0.58) CYP2D6CYP19A1CYP2C9CYP2C19CA12
SCHEMBL14024057 0.77 CYP2A6 (0.58) CYP2D6CYP19A1CYP2C9CYP2C19CA12
SCHEMBL7615000 0.77 TPH1 (0.55) PIM1PIM2
SCHEMBL7615005 0.77 TPH1 (0.55) PIM1PIM2
SCHEMBL21222736 0.75 CYP2A6 (0.55) CYP2D6CYP19A1CYP2C9CYP2C19BRS3
SCHEMBL11541937 0.74 CYP2D6 (0.60) CYP2D6CYP19A1CYP2C9CYP2C19BRS3
SCHEMBL14024068 0.74 HDAC4 (0.42) CYP2D6CYP19A1CYP2C9CYP2C19BRS3
SCHEMBL14025121 0.73 MAPT (0.40) AKT1CDK2MAPTALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1934238-B1 TRIAZOLE COMPOUNDS AND METHODS OF MAKING AND USING THE SAME MELINTA THERAPEUTICS INC (US) 2017-06-28 EP disclosed