Terephthalamide

Terephthalamide

SCHEMBL1906838

N.N.NC(=O)c1ccc(C(N)=O)cc1

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.67
TSHR P16473 2/20 0.67
POLB P06746 1/20 0.67
CYP3A4 P08684 1/20 0.67
MAPT P10636 1/20 0.67
CYP2C19 P33261 1/20 0.67
RECQL P46063 1/20 0.67
BLM P54132 1/20 0.67
PMP22 Q01453 1/20 0.67
HSD17B10 Q99714 1/20 0.67
TDP1 Q9NUW8 1/20 0.67
L3MBTL1 Q9Y468 1/20 0.67
PARP10 Q53GL7 10/20 0.65
PARP4 Q9UKK3 2/20 0.65
PARP15 Q460N3 2/20 0.65
ALDH1A1 P00352 1/20 0.65
KMT2A Q03164 1/20 0.65
PARP14 Q460N5 1/20 0.65
PARP16 Q8N5Y8 1/20 0.65
PARP11 Q9NR21 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Terephthalamide SCHEMBL28199658 1.00 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL23774 0.96 PARP1 (0.71) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL1087289 0.93 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL29102653 0.93 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL27450033 0.93 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL689841 0.93 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL7508927 0.93 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL15328883 0.93 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL11512422 0.93 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT
Terephthalamide SCHEMBL28360111 0.93 PARP1 (0.67) PARP1TSHRPOLBCYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116706004-A Pt-C/composite metal sulfide and preparation method and application thereof 中国科学院苏州纳米技术与纳米仿生研究所 2023-09-05 CN claimed
JP-4683802-B2 2011-05-18 JP claimed
EP-0827976-B1 Polyamide compositions having improved thermal stability SOLVAY ADVANCED POLYMERS LLC (US) 2004-04-07 EP claimed
EP-1198520-B1 METHOD FOR REDUCING MOLD DEPOSIT FORMATION DURING MOLDING OF POLYAMIDES AND COMPOSITION THEREFOR SOLVAY ADVANCED POLYMERS LLC (US) 2003-12-03 EP claimed
US-6531529-B2 Mixture of aromatic polyamide, organohalogen compound and addition polymer SOLVAY ADVANCED POLYMERS, L.L.C. 2003-03-11 US claimed
US-6518341-B1 Reducing mold burning of injection molding formulations comprising impact modified, partially aromatic polyamides containing a copper halide heat stabilizer SOLVAY ADVANCED POLYMERS, LLC 2003-02-11 US claimed
JP-2003503534-A 2003-01-28 JP claimed
EP-1198520-A1 METHOD FOR REDUCING MOLD DEPOSIT FORMATION DURING MOLDING OF POLYAMIDES AND COMPOSITION THEREFOR Solvay Advanced Polymers, LLC (US) 2002-04-24 EP claimed
US-20010053819-A1 Flame retardant anti-drip polyamide compositions SOLVAY ADVANCED POLYMERS, LLC 2001-12-20 US claimed
US-6207745-B1 COMPOSITION COMPRISING HIGH TEMPERATURE POLYPHTHALAMIDE, HALOGEN-CONTAINING ORGANIC COMPOUND, ANTI-DRIP COMPONENT COMPRISING POLYMER FORMED FROM AT LEAST ONE ETHYLENICALLY UNSATURATED MONOMER AND AT LEAST ONE CARBOXYLIC ACID BP AMOCO CORPORATION 2001-03-27 US claimed
WO-2000078869-A1 METHOD FOR REDUCING MOLD DEPOSIT FORMATION DURING MOLDING OF POLYAMIDES AND COMPOSITION THEREFOR SOLVAY ADVANCED POLYMERS, LLC (US) 2000-12-28 WO claimed
EP-0807665-B1 Flame retardant high temperature polyphthalamides having improved thermal stability BP AMOCO CORP (US) 2000-07-12 EP claimed
EP-0986614-A1 FLAME RETARDANT ANTI-DRIP POLYAMIDE COMPOSITIONS BP AMOCO CORPORATION (US) 2000-03-22 EP claimed
US-5962628-A CONTROLLED ENDCAPPING BP AMOCO CORPORATION (US) 1999-10-05 US claimed
WO-1999040157-A1 FLAME RETARDANT ANTI-DRIP POLYAMIDE COMPOSITIONS BP AMOCO CORPORATION (US) 1999-08-12 WO claimed
US-5773500-A BROMINATED POLYSTYRENE WITH ANTIMONY COMPOUND AND MOLDING, CALCIUM OXIDE, MAGNESIUM OXIDE AND ZINC OXIDE AMOCO CORPORATION (US) 1998-06-30 US claimed
US-5763561-A ALKALI METAL HALIDE AND COPPER(I) HALIDE AMOCO CORPORATION (US) 1998-06-09 US claimed
EP-0827976-A2 Polyamide compositions having improved thermal stability AMOCO CORPORATION (US) 1998-03-11 EP claimed
EP-0807665-A2 Flame retardant high temperature polyphthalamides having improved thermal stability AMOCO CORPORATION (US) 1997-11-19 EP claimed
US-5436294-A Impact modifiers for improved ductility and rigidity AMOCO CORPORATION (US) 1995-07-25 US claimed