SCHEMBL19078917

SCHEMBL19078917

NNc1ccc(F)c(NCc2ccccc2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
HTR6 P50406 1/20 0.49
GAA P10253 2/20 0.43
HTT P42858 1/20 0.42
HSD17B10 Q99714 1/20 0.42
IDO1 P14902 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KCNH3 Q9ULD8 1/20 0.41
GPR68 Q15743 1/20 0.41
BACE1 P56817 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
MAPT P10636 2/20 0.40
CYP3A4 P08684 1/20 0.40
MEN1 O00255 1/20 0.40
PABPC1 P11940 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557221 0.80 HDAC1 (0.56) HDAC1HDAC8HDAC6HTR6GAA
SCHEMBL11512276 0.80 HDAC1 (0.59) HDAC1HDAC8HDAC6GAAHTT
SCHEMBL12684764 0.77 HDAC1 (0.60) HDAC1HDAC8HDAC6GAAHTT
SCHEMBL21999822 0.77 HDAC1 (0.56) HDAC1HDAC8HDAC6HSD17B10GPR68
SCHEMBL5444651 0.77 HDAC1 (0.56) HDAC1HDAC8HDAC6GAAHTT
SCHEMBL4982611 0.75 HSD17B10 (0.59) HDAC1HDAC8HDAC6HSD17B10IDO1
SCHEMBL11513455 0.74 MEN1 (0.66) HTTSMN1; SMN2KCNH3GPR68CA12
SCHEMBL6689330 0.73 LMNA (0.55) HDAC1HDAC8HDAC6GAASMN1; SMN2
SCHEMBL13054791 0.70 SMN1; SMN2 (0.46) HDAC1HDAC8HDAC6HTR6GAA
SCHEMBL4270413 0.70 CYP3A4 (0.69) HTTSMN1; SMN2MAPTCYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10018619-B2 Compounds and method of identifying, synthesizing, optimizing and profiling protein modulators HMI Medical Innovations, LLC (US) 2018-07-10 US disclosed
US-10018619-B2 Compounds and method of identifying, synthesizing, optimizing and profiling protein modulators HMI Medical Innovations, LLC (US) 2018-07-10 US disclosed
US-20170191986-A1 Compounds and Method of Identifying, Synthesizing, Optimizing and Profiling Protein Modulators HMI Medical Innovations, LLC 2017-07-06 US disclosed
US-20170191986-A1 Compounds and Method of Identifying, Synthesizing, Optimizing and Profiling Protein Modulators HMI Medical Innovations, LLC 2017-07-06 US disclosed