SCHEMBL1908374

SCHEMBL1908374

CC[As](CC1CCN(C(=O)OC(C)C)CC1)c1ncnc2c1cnn2-c1ccc(S(C)(=O)=O)cc1F

nearest known ligand 0.71

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 20/20 0.71
CYP2C9 P11712 3/20 0.69
KCNH2 Q12809 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL386157 0.83 GPR119 (1.00) GPR119CYP2C9KCNH2
SCHEMBL390409 0.83 GPR119 (0.87) GPR119CYP2C9KCNH2
SCHEMBL389837 0.82 GPR119 (0.82) GPR119CYP2C9KCNH2
SCHEMBL389323 0.82 GPR119 (1.00) GPR119CYP2C9KCNH2
SCHEMBL29376677 0.82 GPR119 (1.00) GPR119CYP2C9KCNH2
SCHEMBL389125 0.78 GPR119 (0.70) GPR119CYP2C9KCNH2
SCHEMBL391113 0.76 GPR119 (0.80) GPR119CYP2C9KCNH2
SCHEMBL389757 0.75 GPR119 (0.87) GPR119CYP2C9KCNH2
SCHEMBL388014 0.75 GPR119 (0.74) GPR119CYP2C9KCNH2
SCHEMBL12505331 0.74 GPR119 (0.78) GPR119CYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2322157-A1 Composition for the treatment of diabetes and conditions related thereto and for the treatment of conditions ameliorated by increasing a blood GLP-1 level Arena Pharmaceuticals, Inc. (US) 2011-05-18 EP disclosed