SCHEMBL1908461

SCHEMBL1908461

CC(=O)N1C(=O)Cc2cc(-c3ccc(F)cc3)ccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.55
PDE5A O76074 1/20 0.43
CYP11B2 P19099 4/20 0.41
CYP11B1 P15538 3/20 0.41
HDAC3 O15379 3/20 0.37
HDAC1 Q13547 3/20 0.37
HDAC2 Q92769 3/20 0.37
HSD17B3 P37058 3/20 0.36
BMPR1B O00238 1/20 0.36
BMPR1A P36894 1/20 0.36
ACVRL1 P37023 1/20 0.36
ACVR1 Q04771 1/20 0.36
BRD4 O60885 1/20 0.36
BRD2 P25440 1/20 0.36
BRD3 Q15059 1/20 0.36
TRIM24 O15164 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
CTSC P53634 1/20 0.36
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2259375 0.88 NOTUM (0.61) NOTUMPDE5AHSD17B3
SCHEMBL1944443 0.79 NOTUM (0.61) NOTUMPDE5AHSD17B3CTSC
SCHEMBL14866100 0.79 CYP11B2 (0.41) NOTUMCYP11B2CYP11B1HSD17B3BRD4
SCHEMBL6690377 0.77 PDE5A (0.67) NOTUMPDE5AHSD17B3
SCHEMBL4303668 0.76 NOTUM (0.61) NOTUMPDE5A
SCHEMBL29643084 0.76 NOTUM (0.61) NOTUMPDE5AHSD17B3BRD4
SCHEMBL5623740 0.76 NOTUM (0.61) NOTUMPDE5AHSD17B3BRD4
SCHEMBL17022647 0.76 NOTUM (0.61) NOTUMPDE5AHDAC1HSD17B3BRD4
SCHEMBL9045039 0.76 NOTUM (0.61) NOTUMPDE5AHDAC1HSD17B3SCN9A
SCHEMBL248856 0.75 NOTUM (0.56) NOTUMPDE5AHSD17B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed