SCHEMBL19086014

SCHEMBL19086014

CC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2sc(C(=O)Nc3ccccc3)cc2C1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.47
HDAC6 Q9UBN7 2/20 0.45
PRMT5 O14744 6/20 0.40
WDR77 Q9BQA1 6/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPK1 P28482 1/20 0.39
PABPC1 P11940 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
CTSK P43235 1/20 0.39
HCRTR2 O43614 3/20 0.39
KDM1A O60341 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086988 0.88 ADORA1 (0.46) ADORA1HDAC6PRMT5WDR77KMT2A
SCHEMBL19086220 0.84 ADORA1 (0.53) ADORA1HDAC6KMT2AMAPTKDM4E
SCHEMBL19086175 0.82 HDAC6 (0.47) HDAC6PRMT5WDR77KMT2AMAPT
SCHEMBL19086221 0.81 HDAC6 (0.43) ADORA1HDAC6PRMT5WDR77KMT2A
SCHEMBL19085999 0.78 TRPV1 (0.41) PRMT5WDR77KMT2AHCRTR2
SCHEMBL19085981 0.78 TRPV1 (0.41) PRMT5WDR77KMT2AHCRTR2
SCHEMBL19086348 0.78 KDM1A (0.41) HDAC6PRMT5WDR77KMT2AMAPT
SCHEMBL19085990 0.78 BRAF (0.40) HDAC6PRMT5WDR77KMT2AHCRTR2
SCHEMBL19086005 0.77 EGFR (0.42) HDAC6PRMT5WDR77KMT2AHCRTR2
SCHEMBL19086001 0.77 JAK2 (0.40) PRMT5WDR77KMT2AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed