SCHEMBL19086221

SCHEMBL19086221

CC[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CCc2sc(C(=O)NC3CCOCC3)cc2C1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.43
ADORA1 P30542 2/20 0.39
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
PRNP P04156 1/20 0.38
PRMT5 O14744 2/20 0.37
WDR77 Q9BQA1 2/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
PDE7A Q13946 1/20 0.35
ALDH1A1 P00352 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086988 0.84 ADORA1 (0.46) HDAC6ADORA1PRMT5WDR77KMT2A
SCHEMBL19086197 0.83 HDAC6 (0.45) HDAC6NPC1RAB9APRNPPRMT5
SCHEMBL19086220 0.82 ADORA1 (0.53) HDAC6ADORA1KMT2AMEN1MAPT
SCHEMBL19086014 0.81 ADORA1 (0.47) HDAC6ADORA1PRMT5WDR77KMT2A
SCHEMBL19086049 0.78 ROCK2 (0.43) HDAC6PRMT5WDR77
SCHEMBL19086017 0.75 HDAC6 (0.36) HDAC6PRMT5WDR77
SCHEMBL19086200 0.75 HDAC6 (0.48) HDAC6NPC1RAB9APRNPPRMT5
SCHEMBL19086018 0.74 ROCK2 (0.44) HDAC6KMT2A
SCHEMBL19086184 0.71 HDAC6 (0.37) HDAC6NPC1RAB9APRNPPRMT5
SCHEMBL19086206 0.71 HDAC6 (0.38) HDAC6PRMT5WDR77KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed