SCHEMBL19086052

SCHEMBL19086052

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(C(=O)NC3CCN(C)CC3)cc2C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.46
ROCK1 Q13464 2/20 0.46
MAPK14 Q16539 1/20 0.40
DCLK1 O15075 1/20 0.39
PDPK1 O15530 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
CHEK2 O96017 1/20 0.39
PIM1 P11309 1/20 0.39
MAPK1 P28482 1/20 0.39
AXL P30530 1/20 0.39
FLT4 P35916 1/20 0.39
FLT3 P36888 1/20 0.39
MAPK9 P45984 1/20 0.39
CSNK1D P48730 1/20 0.39
IRAK1 P51617 1/20 0.39
RPS6KA3 P51812 1/20 0.39
PRKX P51817 1/20 0.39
NEK4 P51957 1/20 0.39
PRKAA1 Q13131 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086053 0.96 ROCK2 (0.43) ROCK2ROCK1MAPK14DCLK1PDPK1
SCHEMBL19086141 0.95 ROCK2 (0.44) ROCK2ROCK1MAPK14CYP3A4HDAC6
SCHEMBL19086020 0.95 ROCK2 (0.44) ROCK2ROCK1MAPK14CYP3A4HDAC6
SCHEMBL19086051 0.94 ROCK2 (0.48) ROCK2ROCK1MAPK14CYP3A4HDAC6
SCHEMBL19086047 0.94 ROCK2 (0.44) ROCK2ROCK1MAPK14CYP3A4HDAC6
SCHEMBL19086056 0.94 ROCK2 (0.43) ROCK2ROCK1MAPK14CYP3A4HDAC6
SCHEMBL19086049 0.93 ROCK2 (0.43) ROCK2ROCK1MAPK14CYP3A4HDAC6
SCHEMBL19086055 0.92 ROCK2 (0.40) ROCK2ROCK1MAPK14CYP3A4HDAC6
SCHEMBL19086054 0.91 ROCK2 (0.41) ROCK2ROCK1MAPK14CYP3A4HDAC6
SCHEMBL19086046 0.91 ROCK2 (0.41) ROCK2ROCK1MAPK14CYP3A4HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed