SCHEMBL19086578

SCHEMBL19086578

Cn1c(=O)c(C(=O)NNCC(=O)O)c(O)c2cc(C(=O)NC(c3ccccc3)c3ccccc3)ccc21

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 7/20 0.60
L3MBTL1 Q9Y468 1/20 0.50
MEN1 O00255 7/20 0.48
KMT2A Q03164 7/20 0.48
NLRP3 Q96P20 2/20 0.48
GAA P10253 1/20 0.47
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
EGLN1 Q9GZT9 1/20 0.44
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GSK3B P49841 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17578433 0.90 HIF1A (0.72) HIF1AL3MBTL1MEN1KMT2ANPC1
SCHEMBL19086545 0.83 HIF1A (0.52) HIF1AL3MBTL1MEN1KMT2ANLRP3
SCHEMBL23953030 0.81 HIF1A (0.48) HIF1AL3MBTL1MEN1KMT2ANLRP3
SCHEMBL17578572 0.75 HIF1A (1.00) HIF1AMEN1KMT2ANPC1RAB9A
SCHEMBL19086553 0.71 HPGDS (0.46) MEN1KMT2AGAAKDM4E
SCHEMBL2383791 0.70 HIF1A (0.72) HIF1AMEN1KMT2ANPC1RAB9A
SCHEMBL17578567 0.69 HIF1A (0.67) HIF1AMEN1KMT2ANPC1RAB9A
SCHEMBL2382524 0.69 HIF1A (0.61) HIF1AEGLN1
SCHEMBL2399702 0.69 MEN1 (0.77) HIF1AL3MBTL1MEN1KMT2ANPC1
SCHEMBL2383420 0.69 HIF1A (0.69) HIF1AEGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3190104-B1 QUINOLINONE COMPOUND AND USE THEREOF SUNSHINE LAKE PHARMA CO LTD (CN) 2021-10-27 EP disclosed
EP-3190104-A1 QUINOLINONE COMPOUND AND USE THEREOF Sunshine Lake Pharma Co., Ltd. (CN) 2017-07-12 EP disclosed