SCHEMBL19089030

SCHEMBL19089030

Cc1nc2c(F)cc(-c3nc(Nc4ccc5c(n4)CCN(CCS(C)(=O)=NC#N)C5)nc(CN(C)CCN4CCc5nc(Nc6ncc(F)c(-c7cc(F)c8nc(C)n([C@H]9CC[C@H](C)CC9)c8c7)n6)ccc5C4)c3F)cc2n1C(C)C

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.76
CDK2 P24941 20/20 0.76
CDK6 Q00534 20/20 0.76
CDK1 P06493 7/20 0.76
CDK7 P50613 7/20 0.76
CDK9 P50750 7/20 0.76
CDK5 Q00535 7/20 0.76
CCNA2 P20248 13/20 0.66
CCND3 P30281 13/20 0.66
CHEK1 O14757 1/20 0.61
CCNT1 O60563 1/20 0.61
JAK2 O60674 1/20 0.61
CHEK2 O96017 1/20 0.61
EGFR P00533 1/20 0.61
RAF1 P04049 1/20 0.61
NTRK1 P04629 1/20 0.61
PDGFRB P09619 1/20 0.61
SRC P12931 1/20 0.61
CCNB1 P14635 1/20 0.61
BRAF P15056 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19088988 0.87 CDK4 (1.00) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19089002 0.81 CDK4 (0.88) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19088996 0.81 CDK4 (1.00) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19089031 0.79 CDK4 (0.85) CDK4CDK2CDK6CDK1CDK7
SCHEMBL17485308 0.79 CDK4 (0.83) CDK4CDK2CDK6CDK1CDK7
SCHEMBL31066529 0.78 CDK4 (0.88) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19089443 0.78 CDK4 (0.88) CDK4CDK2CDK6CDK1CDK7
SCHEMBL29839750 0.78 CDK4 (1.00) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19089039 0.78 CDK4 (1.00) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19089096 0.78 CDK4 (0.81) CDK4CDK2CDK6CDK1CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114512-A1 NITROGEN-CONTAINING FUSED HETEROCYCLIC COMPOUND, AS WELL AS PREPARATION METHOD, INTERMEDIATE, COMPOSITION AND APPLICATION THEREOF 上海医药集团股份有限公司 2017-07-06 WO disclosed