SCHEMBL19098724

SCHEMBL19098724

Cn1nccc1Nc1nccc(-c2ccc(NC(=O)Cc3ccccc3)c(C#N)c2)n1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 1/20 0.52
MAPK1 P28482 18/20 0.52
IKBKB O14920 1/20 0.45
MAPK6 Q16659 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19099170 0.92 MAP3K14 (0.49) MAP3K14MAPK1
SCHEMBL19098731 0.89 MAPK1 (0.55) MAP3K14MAPK1MAPK6
SCHEMBL19099029 0.89 MAPK1 (0.58) MAP3K14MAPK1
SCHEMBL19098869 0.88 MAPK1 (0.53) MAPK1IKBKBMAPK6
SCHEMBL19099153 0.87 MAPK1 (0.54) MAPK1
SCHEMBL19098889 0.87 MAPK1 (0.52) MAPK1IKBKBMAPK6
SCHEMBL19099039 0.86 MAPK1 (0.57) MAP3K14MAPK1
SCHEMBL19099169 0.84 MAPK1 (0.59) MAP3K14MAPK1MAPK6
SCHEMBL19099027 0.84 MAPK1 (0.58) MAP3K14MAPK1MAPK6
SCHEMBL19098885 0.83 IKBKB (0.63) MAPK1IKBKBMAPK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922405-B Compound with ERK kinase inhibitory activity, preparation method and application thereof 中国科学院上海药物研究所 2021-02-19 CN disclosed
WO-2017114510-A1 COMPOUND HAVING ERK KINASE INHIBITORY ACTIVITY, METHOD FOR PREPARATION THEREOF, AND USE THEREOF 中国科学院上海药物研究所 2017-07-06 WO disclosed