SCHEMBL19099039

SCHEMBL19099039

Cn1nccc1Nc1nccc(-c2ccc(NC(=O)Cc3cccnc3Cl)c(C#N)c2)n1

nearest known ligand 0.57

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 19/20 0.57
MAP3K14 Q99558 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19098731 0.92 MAPK1 (0.55) MAPK1MAP3K14
SCHEMBL19099169 0.89 MAPK1 (0.59) MAPK1MAP3K14
SCHEMBL19099029 0.88 MAPK1 (0.58) MAPK1MAP3K14
SCHEMBL19098724 0.86 MAP3K14 (0.52) MAPK1MAP3K14
SCHEMBL19099027 0.86 MAPK1 (0.58) MAPK1MAP3K14
SCHEMBL19099170 0.85 MAP3K14 (0.49) MAPK1MAP3K14
SCHEMBL19099165 0.80 MAPK1 (0.82) MAPK1
SCHEMBL19099032 0.80 MAPK1 (0.55) MAPK1
SCHEMBL19099286 0.79 MAPK1 (0.62) MAPK1MAP3K14
SCHEMBL19099172 0.79 MAPK1 (0.62) MAPK1MAP3K14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922405-B Compound with ERK kinase inhibitory activity, preparation method and application thereof 中国科学院上海药物研究所 2021-02-19 CN disclosed
WO-2017114510-A1 COMPOUND HAVING ERK KINASE INHIBITORY ACTIVITY, METHOD FOR PREPARATION THEREOF, AND USE THEREOF 中国科学院上海药物研究所 2017-07-06 WO disclosed