SCHEMBL19112978

SCHEMBL19112978

CC(C)(C)NCC(=O)N1CCC(CNC(=O)c2cc(C(F)(F)F)cc(C(F)(F)P)c2)CC1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.58
CACNA1I Q9P0X4 7/20 0.58
MCHR1 Q99705 3/20 0.42
RORC P51449 1/20 0.42
CCR2 P41597 1/20 0.42
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA1A P35348 1/20 0.41
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1428162 0.95 KCNH2 (0.64) KCNH2CACNA1IMCHR1KDM4EPKM
SCHEMBL4277516 0.89 KCNH2 (0.57) KCNH2CACNA1IKDM4EPKM
SCHEMBL19113096 0.83 KCNH2 (0.60) KCNH2CACNA1IRORCCCR2
SCHEMBL19113176 0.82 KCNH2 (0.58) KCNH2CACNA1IMCHR1RORCCCR2
SCHEMBL4278214 0.81 KCNH2 (0.59) KCNH2CACNA1IMCHR1RORCCCR2
SCHEMBL20056079 0.80 KCNH2 (0.62) KCNH2CACNA1IMCHR1RORCCCR2
SCHEMBL1432591 0.80 KCNH2 (0.62) KCNH2CACNA1IMCHR1RORCCCR2
SCHEMBL19113450 0.80 KCNH2 (0.53) KCNH2CACNA1IMCHR1RORCCCR2
SCHEMBL4271541 0.80 KCNH2 (0.57) KCNH2CACNA1IMCHR1RORCCCR2
SCHEMBL13569703 0.80 KCNH2 (0.46) KCNH2CACNA1IRORCCCR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3189839-A1 N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS Taro Pharmaceuticals Inc. (CA) 2017-07-12 EP disclosed