SCHEMBL19119376

SCHEMBL19119376

CN(Cc1nsc(NC(=O)NCc2cccc(F)c2)n1)C(=O)O.N#CC1CC1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.45
ROCK1 Q13464 2/20 0.45
ATG4B Q9Y4P1 1/20 0.41
NPC1 O15118 1/20 0.39
NAMPT P43490 3/20 0.38
EPHX2 P34913 1/20 0.38
AURKA O14965 1/20 0.37
CDK8 P49336 1/20 0.37
AURKB Q96GD4 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PAX8 Q06710 1/20 0.36
NLRP3 Q96P20 1/20 0.36
ANPEP P15144 1/20 0.36
MAPT P10636 3/20 0.36
TP53 P04637 2/20 0.36
POLB P06746 1/20 0.36
LMNA P02545 1/20 0.35
CPS1 P31327 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19119463 0.91 ROCK2 (0.48) ROCK2ROCK1ATG4BNPC1NAMPT
Cyclohexane SCHEMBL19119453 0.90 ROCK2 (0.50) ROCK2ROCK1ATG4BNPC1NAMPT
Cyclopentane SCHEMBL19119283 0.90 ROCK2 (0.50) ROCK2ROCK1ATG4BNPC1NAMPT
SCHEMBL19119284 0.88 ROCK2 (0.45) ROCK2ROCK1ATG4BNPC1NAMPT
SCHEMBL19119378 0.86 ROCK2 (0.44) ROCK2ROCK1ATG4BNPC1NAMPT
SCHEMBL19119492 0.85 ROCK2 (0.43) ROCK2ROCK1ATG4BNPC1NAMPT
SCHEMBL354384 0.83 ROCK2 (0.46) ROCK2ROCK1ATG4BNPC1NAMPT
SCHEMBL354401 0.83 ROCK2 (0.47) ROCK2ROCK1ATG4BNPC1NAMPT
SCHEMBL354589 0.82 ROCK2 (0.47) ROCK2ROCK1ATG4BNPC1NAMPT
SCHEMBL352913 0.81 ROCK2 (0.48) ROCK2ROCK1ATG4BNPC1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200440-B1 ANTIBACTERIAL AMIDE AND SULFONAMIDE SUBSTITUTED HETEROCYCLIC UREA COMPOUNDS CRESTONE INC (US) 2017-07-19 EP claimed