SCHEMBL19119447

SCHEMBL19119447

CN(Cc1csc(NC(=O)NCc2cccc(F)c2)n1)C(=O)Oc1cnn2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 13/20 0.47
ROCK2 O75116 13/20 0.47
ATG4B Q9Y4P1 1/20 0.40
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NAMPT P43490 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL353239 0.88 ROCK2 (0.48) ROCK1ROCK2ATG4BKDM4ENPC1
SCHEMBL19119209 0.85 ROCK1 (0.48) ROCK1ROCK2ATG4B
SCHEMBL19119187 0.85 ROCK1 (0.48) ROCK1ROCK2ATG4BNAMPT
SCHEMBL19119394 0.84 ROCK1 (0.47) ROCK1ROCK2ATG4BNAMPT
SCHEMBL19119288 0.84 ROCK1 (0.46) ROCK1ROCK2ATG4BKDM4EALDH1A1
SCHEMBL19119102 0.83 ROCK1 (0.48) ROCK1ROCK2ATG4B
SCHEMBL19119292 0.83 ROCK2 (0.51) ROCK1ROCK2ATG4BNAMPT
SCHEMBL19119499 0.82 ROCK1 (0.50) ROCK1ROCK2ATG4B
SCHEMBL19118736 0.82 ROCK1 (0.48) ROCK1ROCK2ATG4B
SCHEMBL19119346 0.82 ROCK1 (0.49) ROCK1ROCK2ATG4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200440-B1 ANTIBACTERIAL AMIDE AND SULFONAMIDE SUBSTITUTED HETEROCYCLIC UREA COMPOUNDS CRESTONE INC (US) 2017-07-19 EP claimed