SCHEMBL19119503

SCHEMBL19119503

CN(Cc1csc(NC(=O)NCc2cccc(F)c2)n1)C(=O)Oc1cc(O)nnc1Cl

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 16/20 0.49
ROCK2 O75116 15/20 0.49
EPHX2 P34913 1/20 0.40
HSD17B13 Q7Z5P4 1/20 0.40
ATG4B Q9Y4P1 1/20 0.39
SGK1 O00141 1/20 0.39
AKT1 P31749 1/20 0.39
GSK3B P49841 1/20 0.39
LIMK1 P53667 1/20 0.39
TNK2 Q07912 1/20 0.39
DMPK Q09013 1/20 0.39
MYLK Q15746 1/20 0.39
CDC42BPA Q5VT25 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19119156 0.93 ROCK1 (0.49) ROCK1ROCK2EPHX2HSD17B13ATG4B
SCHEMBL19119113 0.91 ROCK2 (0.47) ROCK1ROCK2EPHX2ATG4B
SCHEMBL352559 0.87 ROCK2 (0.50) ROCK1ROCK2EPHX2HSD17B13ATG4B
SCHEMBL19119187 0.84 ROCK1 (0.48) ROCK1ROCK2EPHX2ATG4B
SCHEMBL19119157 0.83 ROCK1 (0.51) ROCK1ROCK2ATG4BSGK1AKT1
SCHEMBL19119292 0.83 ROCK2 (0.51) ROCK1ROCK2EPHX2ATG4B
SCHEMBL19118770 0.83 ROCK2 (0.49) ROCK1ROCK2EPHX2HSD17B13ATG4B
SCHEMBL19119270 0.83 ROCK2 (0.50) ROCK1ROCK2EPHX2ATG4B
SCHEMBL19118739 0.82 ROCK1 (0.51) ROCK1ROCK2ATG4BSGK1AKT1
SCHEMBL19119382 0.82 ROCK1 (0.48) ROCK1ROCK2EPHX2ATG4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200440-B1 ANTIBACTERIAL AMIDE AND SULFONAMIDE SUBSTITUTED HETEROCYCLIC UREA COMPOUNDS CRESTONE INC (US) 2017-07-19 EP claimed