SCHEMBL1912766

SCHEMBL1912766

CCCCn1c(-c2ccccc2)nc(C#N)c1CO

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.51
HSD17B10 Q99714 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
NR1H3 Q13133 1/20 0.43
PDE4B Q07343 4/20 0.41
GRK6 P43250 1/20 0.39
TP53 P04637 2/20 0.38
HSD11B1 P28845 2/20 0.38
MEN1 O00255 2/20 0.38
ALOX15 P16050 2/20 0.38
CASP1 P29466 2/20 0.38
KMT2A Q03164 2/20 0.38
SAE1 Q9UBE0 2/20 0.38
UBA2 Q9UBT2 2/20 0.38
NSD2 O96028 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
HSP90AA1 P07900 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL652738 0.85 TSHR (0.58) TSHRHSD17B10KDM4EALDH1A1HPGD
SCHEMBL648785 0.81 TSHR (0.56) TSHRHSD17B10KDM4EALDH1A1HPGD
SCHEMBL11095759 0.80 TSHR (0.55) TSHRHSD17B10KDM4EALDH1A1HPGD
SCHEMBL647960 0.80 TSHR (0.55) TSHRHSD17B10KDM4EALDH1A1HPGD
SCHEMBL650051 0.80 TSHR (0.55) TSHRHSD17B10KDM4EALDH1A1HPGD
SCHEMBL1912781 0.79 TSHR (0.50) TSHRHSD17B10KDM4EALDH1A1HPGD
SCHEMBL1912780 0.77 TSHR (0.51) TSHRHSD17B10KDM4EALDH1A1HPGD
SCHEMBL649593 0.75 TSHR (0.52) TSHRHSD17B10KDM4EALDH1A1HPGD
SCHEMBL11092583 0.74 TSHR (0.51) TSHRHSD17B10KDM4EALDH1A1HPGD
SCHEMBL6619406 0.74 TSHR (0.58) TSHRHSD17B10KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119665-B2 Aryl imidazoles and related compounds as C5a receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-02-21 US disclosed
US-8119665-B2 Aryl imidazoles and related compounds as C5a receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-02-21 US disclosed
US-7186734-B2 Aryl imidazoles and related compounds as C5a receptor modulators NEUROGEN CORPORATION (US) 2007-03-06 US disclosed
US-7186734-B2 Aryl imidazoles and related compounds as C5a receptor modulators NEUROGEN CORPORATION (US) 2007-03-06 US disclosed