SCHEMBL19129148

SCHEMBL19129148

CC(C)[C@H](NC(=O)CN1CC2(CCCN2C(=O)OCc2ccccc2)C1=O)C(N)=O

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IL1RN P18510 1/20 0.42
ERAP2 Q6P179 1/20 0.42
ERAP1 Q9NZ08 1/20 0.42
ELANE P08246 7/20 0.39
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSK P43235 1/20 0.38
CTRC Q99895 2/20 0.38
LMNA P02545 1/20 0.38
ECE1 P42892 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15937101 0.94 GRIN2B (0.41) IL1RNERAP2ERAP1ELANECTSL
SCHEMBL17351809 0.94 GRIN2B (0.41) IL1RNERAP2ERAP1ELANECTSL
SCHEMBL15937244 0.91 IL1RN (0.36) IL1RNERAP2ERAP1LMNA
SCHEMBL20126641 0.91 IL1RN (0.36) IL1RNERAP2ERAP1LMNA
SCHEMBL17351899 0.91 IL1RN (0.36) IL1RNERAP2ERAP1LMNA
SCHEMBL19129091 0.86 GRIN2B (0.37) ELANELMNA
SCHEMBL15937085 0.86 CCR1 (0.40) IL1RNERAP2ERAP1CTSLCTSB
SCHEMBL17356203 0.85 ALDH1A1 (0.39)
SCHEMBL17359168 0.83 CYP2C19 (0.42)
SCHEMBL20126625 0.82 GRIN2B (0.39) ELANELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9708335-B2 Spiro-lactam NMDA receptor modulators and uses thereof Apytinyx Inc. (US) 2017-07-18 US disclosed
US-9708335-B2 Spiro-lactam NMDA receptor modulators and uses thereof Apytinyx Inc. (US) 2017-07-18 US disclosed