SCHEMBL19149201

SCHEMBL19149201

N#CC([C@@H](C1CCCC1)n1cc(-c2ncnc3[nH]ccc23)cn1)P(=O)(O)O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 17/20 0.71
JAK1 P23458 14/20 0.71
JAK3 P52333 5/20 0.71
TYK2 P29597 4/20 0.71
DAPK3 O43293 2/20 0.65
PAK4 O96013 2/20 0.65
ABL1 P00519 2/20 0.65
RET P07949 2/20 0.65
LTK P29376 2/20 0.65
CSNK1A1 P48729 2/20 0.65
CLK2 P49760 2/20 0.65
TNK2 Q07912 2/20 0.65
ROCK1 Q13464 2/20 0.65
DYRK1A Q13627 2/20 0.65
IKBKE Q14164 2/20 0.65
NTRK3 Q16288 2/20 0.65
NTRK2 Q16620 2/20 0.65
LRRK2 Q5S007 2/20 0.65
TAOK1 Q7L7X3 2/20 0.65
CAMK1D Q8IU85 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1612829 0.86 JAK2 (0.70) JAK2JAK1JAK3TYK2DAPK3
Ruxolitinib SCHEMBL29357426 0.83 JAK2 (1.00) JAK2JAK1JAK3TYK2DAPK3
Ruxolitinib SCHEMBL31073616 0.83 JAK2 (1.00) JAK2JAK1JAK3TYK2DAPK3
Ruxolitinib SCHEMBL1369365 0.83 JAK2 (1.00) JAK2JAK1JAK3TYK2DAPK3
Ruxolitinib SCHEMBL1371422 0.83 JAK2 (1.00) JAK2JAK1JAK3TYK2DAPK3
Ruxolitinib SCHEMBL29677819 0.83 JAK2 (1.00) JAK2JAK1JAK3TYK2DAPK3
SCHEMBL1610290 0.81 JAK2 (0.68) JAK2JAK1JAK3TYK2DAPK3
Phosphoric Acid SCHEMBL3008015 0.80 JAK2 (0.68) JAK2JAK1JAK3TYK2DAPK3
Phosphoric Acid SCHEMBL30338770 0.80 JAK2 (0.68) JAK2JAK1JAK3TYK2DAPK3
Phosphoric Acid SCHEMBL20474415 0.79 JAK2 (0.93) JAK2JAK1JAK3TYK2DAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017125097-A1 CRYSTALLINE FORMS OF (3R)-3-CYCLOPENTYL-3-[4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4- YL)PYRAZOL-L-YL]PROPANENITRILE SALTS AND PREPARATION THEREOF ZENTIVA, K.S. (CZ) 2017-07-27 WO disclosed