SCHEMBL1915239

SCHEMBL1915239

COc1cccc2ccc(C=O)nc12

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.57
CCR1 P32246 1/20 0.57
KMT2A Q03164 9/20 0.56
MAPT P10636 3/20 0.56
ALDH1A1 P00352 2/20 0.56
HPGD P15428 2/20 0.56
KDM4E B2RXH2 1/20 0.56
GLA P06280 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
MEN1 O00255 7/20 0.50
NPC1 O15118 4/20 0.50
RAB9A P51151 4/20 0.50
ECE2 P0DPD6 1/20 0.49
AGTR1 P30556 2/20 0.48
PDE10A Q9Y233 1/20 0.47
POLB P06746 2/20 0.45
OPRK1 P41145 1/20 0.45
F2R P25116 1/20 0.43
NQO2 P16083 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29694483 1.00 MCHR1 (0.57) MCHR1CCR1KMT2AMAPTALDH1A1
SCHEMBL13739153 0.82 MCHR1 (0.60) MCHR1CCR1KMT2AMAPTALDH1A1
SCHEMBL27947067 0.82 NCF1 (0.48) MCHR1CCR1MAPTALDH1A1HPGD
SCHEMBL16107146 0.80 MCHR1 (0.54) MCHR1KMT2AMAPTALDH1A1HPGD
SCHEMBL12066587 0.79 KMT2A (0.62) MCHR1KMT2AMAPTALDH1A1HPGD
SCHEMBL7513556 0.79 KMT2A (0.62) MCHR1KMT2AMAPTALDH1A1HPGD
SCHEMBL28613689 0.79 MCHR1 (0.63) MCHR1CCR1KMT2AMAPTKDM4E
SCHEMBL7513553 0.79 KMT2A (0.62) MCHR1KMT2AMAPTALDH1A1HPGD
SCHEMBL763980 0.79 CCR1 (0.47) MCHR1CCR1KMT2AMAPTALDH1A1
SCHEMBL13739010 0.78 MCHR1 (0.66) MCHR1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 94 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119529141-A Preparation method of quinoline amino binuclear metal titanium zirconium hafnium catalyst and application of catalyst in olefin polymerization 青岛科技大学 2025-02-28 CN disclosed
US-20240010913-A1 RED FLUORESCENT SENSOR COMPOUNDS FOR THE DETECTION OF METAL IONS FEMTONICS KFT. (HU) 2024-01-11 US disclosed
WO-2022118054-A1 RED FLUORESCENT SENSOR COMPOUNDS FOR THE DETECTION OF METAL IONS FEMTONICS KFT. (HU) 2022-06-09 WO disclosed
EP-3318561-B1 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC (US) 2021-12-22 EP disclosed
EP-3318561-B1 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC (US) 2021-12-22 EP disclosed
WO-2021008588-A1 CLASS OF PYRIMIDINE QUINOLINE DERIVATIVES AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 广州新民培林医药科技有限公司 2021-01-21 WO disclosed
US-10813939-B2 Bromodomain inhibitor as adjuvant in cancer immunotherapy H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2020-10-27 US disclosed
US-10676484-B2 Compositions and methods for treating leukemia DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-06-09 US disclosed
US-20200148702-A1 COMPOSITIONS AND METHODS FOR TREATING NEOPLASIA, INFLAMMATORY DISEASE AND OTHER DISORDERS DANA FARBER CANCER INST INC (US) 2020-05-14 US disclosed
US-10562916-B2 Substituted quinoxalines as PDE-10 inhibitors SUNOVION PHARMACEUTICALS, INC. (US) 2020-02-18 US disclosed
WO-2011150156-A2 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2011-12-01 WO disclosed
WO-2011079274-A1 AMINOPYRIMIDINE KINASE INHIBITORS Jasco Pharmaceuticals, LLC (US) 2011-06-30 WO disclosed
US-20110152235-A1 Aminopyrimidine Kinase Inhibitors Jasco Pharmaceuticals, LLC (US) 2011-06-23 US disclosed
WO-2010132615-A1 HYDRAZONE COMPOUNDS AND THEIR USE STEIN PHILIP (US) 2010-11-18 WO disclosed
US-20070173525-A1 Tyrosine kinase inhibitors MERCK SHARP & DOHME CORP. 2007-07-26 US disclosed
EP-1496897-A4 TYROSINE KINASE INHIBITORS MERCK & CO INC (US) 2006-05-10 EP disclosed
US-20050239815-A1 Tyrosine kinase inhibitors KIM ANNETTE J 2005-10-27 US disclosed
EP-1496897-A1 TYROSINE KINASE INHIBITORS Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2003086395-A1 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2003-10-23 WO disclosed
US-3953428-A ANTIBACTERIAL YAMANOUCHI PHARMACEUTICAL CO., LTD. (JA) 1976-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070173525-A1 Tyrosine kinase inhibitors ABL1, JAK2, ERBB2 MCHR1 417/4885CCR1 2228/4885KMT2A 687/4885
US-20050239815-A1 Tyrosine kinase inhibitors ABL1, JAK2, ERBB2 MCHR1 417/4885CCR1 2228/4885KMT2A 687/4885
US-10813939-B2 Bromodomain inhibitor as adjuvant in cancer immunotherapy BRDT, BRD4, BRD1 MCHR1 4238/4885CCR1 205/4885KMT2A 415/4885
US-10676484-B2 Compositions and methods for treating leukemia MCL1, ABL1, FLT3 MCHR1 3842/4885CCR1 128/4885KMT2A 231/4885
US-20240010913-A1 RED FLUORESCENT SENSOR COMPOUNDS FOR THE DETECTION OF METAL IONS SLC30A6, SLC30A7, SLC39A14 MCHR1 909/4885CCR1 3740/4885KMT2A 3909/4885
US-10562916-B2 Substituted quinoxalines as PDE-10 inhibitors PDE4A, PDE2A, PDE9A MCHR1 3827/4885CCR1 3552/4885KMT2A 1967/4885
US-20200148702-A1 COMPOSITIONS AND METHODS FOR TREATING NEOPLASIA, INFLAMMATORY DISEASE AND OTHER DISORDERS BRPF3, EP300, BRD3 MCHR1 4735/4885CCR1 1459/4885KMT2A 134/4885
US-20110152235-A1 Aminopyrimidine Kinase Inhibitors PIM1, PIM2, PIM3 MCHR1 4221/4885CCR1 2856/4885KMT2A 1400/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.