SCHEMBL1918932

SCHEMBL1918932

CNC(=O)c1c(-c2ccc(F)cc2)oc2cc(NS(=O)(=O)CCCO)c(-c3cccc(C(=O)N(c4ccccn4)C4CC4)c3)cc12

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.41
CYP2C8 P10632 2/20 0.41
KCNH2 Q12809 2/20 0.41
NR1I2 O75469 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1918583 0.91 CYP3A4 (0.39) CYP3A4CYP2C8
SCHEMBL1918518 0.91 CYP3A4 (0.41) CYP3A4KCNH2
SCHEMBL1918933 0.85
SCHEMBL1919012 0.83 CYP3A4 (0.42) CYP3A4CYP2C8
SCHEMBL2142748 0.83 CYP2C8 (0.62) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL1919314 0.82 CYP3A4 (0.40) CYP3A4CYP2C8KCNH2
SCHEMBL1920430 0.82 CYP2C8 (0.46) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL14323750 0.82 CYP3A4 (0.44) CYP3A4CYP2C8
SCHEMBL2431623 0.81 ALDH1A1 (0.45) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL2141940 0.80 CYP3A4 (0.40) CYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545042-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP disclosed
WO-2011112191-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed
EP-2326633-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2011-06-01 EP disclosed
WO-2010030592-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2010-03-18 WO disclosed