SCHEMBL19189869

SCHEMBL19189869

Fc1cccnc1C1CCC(c2nnc3n2-c2ccc(Cl)cc2COC3)CC1

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 19/20 0.66
KCNH2 Q12809 7/20 0.51
AVPR2 P30518 5/20 0.51
OXTR P30559 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14853323 1.00 AVPR1A (0.66) AVPR1AKCNH2AVPR2OXTR
SCHEMBL14844441 1.00 AVPR1A (0.66) AVPR1AKCNH2AVPR2OXTR
SCHEMBL2539944 0.84 AVPR1A (0.66) AVPR1AKCNH2AVPR2
SCHEMBL2540655 0.84 AVPR1A (0.66) AVPR1AKCNH2AVPR2
SCHEMBL2539946 0.84 AVPR1A (0.66) AVPR1AKCNH2AVPR2
SCHEMBL19189883 0.84 AVPR1A (0.65) AVPR1AKCNH2AVPR2OXTR
SCHEMBL2542010 0.83 AVPR1A (0.67) AVPR1AKCNH2AVPR2
SCHEMBL2542009 0.83 AVPR1A (0.67) AVPR1AKCNH2AVPR2
SCHEMBL2546578 0.83 AVPR1A (0.67) AVPR1AKCNH2AVPR2
SCHEMBL5102063 0.82 AVPR1A (0.80) AVPR1AKCNH2AVPR2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763997-B1 CYCLOHEXYL-4H,6H-5-OXA-2,3,10B-TRIAZA-BENZO[E]AZULENES AS V1A ANTAGONISTS HOFFMANN LA ROCHE (CH) 2017-08-02 EP disclosed