SCHEMBL19189883

SCHEMBL19189883

FC1CCC(c2nnc3n2-c2ccc(Cl)cc2COC3)CC1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 20/20 0.65
KCNH2 Q12809 8/20 0.53
AVPR2 P30518 4/20 0.48
OXTR P30559 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20382772 0.89 AVPR1A (0.66) AVPR1AKCNH2AVPR2
SCHEMBL5094961 0.87 AVPR1A (0.64) AVPR1AKCNH2AVPR2OXTR
SCHEMBL14853325 0.86 AVPR1A (0.58) AVPR1AKCNH2AVPR2
SCHEMBL14844173 0.86 AVPR1A (0.58) AVPR1AKCNH2AVPR2
SCHEMBL14801823 0.85 AVPR1A (0.60) AVPR1AKCNH2AVPR2OXTR
SCHEMBL14801989 0.85 AVPR1A (0.60) AVPR1AKCNH2AVPR2OXTR
SCHEMBL14853323 0.84 AVPR1A (0.66) AVPR1AKCNH2AVPR2OXTR
SCHEMBL14844441 0.84 AVPR1A (0.66) AVPR1AKCNH2AVPR2OXTR
SCHEMBL19189869 0.84 AVPR1A (0.66) AVPR1AKCNH2AVPR2OXTR
SCHEMBL14844408 0.84 AVPR1A (0.60) AVPR1AKCNH2AVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763997-B1 CYCLOHEXYL-4H,6H-5-OXA-2,3,10B-TRIAZA-BENZO[E]AZULENES AS V1A ANTAGONISTS HOFFMANN LA ROCHE (CH) 2017-08-02 EP disclosed