SCHEMBL19192050

SCHEMBL19192050

CN[C@@]12CCC[C@@](NC(=O)c3cccc(Cl)c3)(CC1)C2

nearest known ligand 0.70

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 10/20 0.70
FPR2 P25090 8/20 0.70
IDO1 P14902 6/20 0.52
TP53 P04637 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19192366 0.86 FPR2 (0.76) GRM5FPR2NPC1RAB9A
SCHEMBL19192151 0.86 FPR2 (0.76) GRM5FPR2NPC1RAB9A
SCHEMBL11027368 0.84 GRM5 (0.66) GRM5FPR2IDO1L3MBTL1
SCHEMBL9960986 0.84 GRM5 (0.62) GRM5FPR2IDO1TP53L3MBTL1
SCHEMBL11028972 0.84 GRM5 (0.62) GRM5FPR2IDO1TP53L3MBTL1
SCHEMBL11028870 0.84 GRM5 (0.62) GRM5FPR2IDO1TP53L3MBTL1
SCHEMBL11030302 0.83 GRM5 (0.67) GRM5FPR2IDO1TP53
SCHEMBL19192385 0.83 GRM5 (1.00) GRM5FPR2IDO1
SCHEMBL10151943 0.83 GRM5 (1.00) GRM5FPR2IDO1
SCHEMBL11029977 0.82 GRM5 (0.73) GRM5FPR2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2654422-B1 Bicyclo[3.2.1]octyl amide derivatives as allosteric modulators of the metabotropic glutamate receptor 5 (mGlu5 or mGluR5) for the treatment of central nervous system (CNS) disorders H LUNDBECK AS (DK) 2017-08-02 EP disclosed