SCHEMBL19199529

SCHEMBL19199529

CCN(CC1CCCC1)c1nc2ccccc2cc1CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)/C(N)=N/N(C)N

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.34
GPBAR1 Q8TDU6 4/20 0.33
BACE1 P56817 1/20 0.33
SGMS1 Q86VZ5 1/20 0.31
SGMS2 Q8NHU3 1/20 0.31
BCHE P06276 1/20 0.30
ACHE P22303 1/20 0.30
SIGMAR1 Q99720 1/20 0.30
CETP P11597 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19188648 0.97 TACR1 (0.34) TACR1GPBAR1SIGMAR1CETPTRPM8
SCHEMBL19188494 0.93 TACR1 (0.34) TACR1GPBAR1BACE1SIGMAR1CETP
SCHEMBL5624904 0.90 GPBAR1 (0.35) TACR1GPBAR1BACE1BCHEACHE
SCHEMBL19188677 0.89 GPBAR1 (0.35) TACR1GPBAR1BACE1BCHEACHE
SCHEMBL14602924 0.89 GPBAR1 (0.38) TACR1GPBAR1BACE1CETPTRPM8
SCHEMBL19189353 0.88 TACR1 (0.34) TACR1GPBAR1BACE1SGMS1SGMS2
SCHEMBL16743088 0.85 CRHR1 (0.33) TACR1GPBAR1BACE1BCHEACHE
SCHEMBL5623760 0.85 GPBAR1 (0.34) TACR1GPBAR1BACE1BCHEACHE
SCHEMBL19188694 0.85 TACR1 (0.34) TACR1GPBAR1BACE1SGMS1SGMS2
SCHEMBL19189308 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848430-B1 NOVEL BENZYLAMINE DERIVATIVES AS CETP INHIBITORS Dr Reddys Laboratories Ltd (IN) 2017-08-02 EP disclosed