SCHEMBL19199863

SCHEMBL19199863

O=C(c1cc(Cn2c(=O)[nH]c(=O)c3ccccc32)ccc1F)N1CCN(CC(F)(F)F)CC1

nearest known ligand 0.79

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.79
PARP2 Q9UGN5 19/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19200039 0.90 PARP1 (0.65) PARP1PARP2
SCHEMBL19200808 0.89 PARP1 (0.78) PARP1PARP2
SCHEMBL29568133 0.89 PARP1 (0.75) PARP1PARP2
SCHEMBL19200137 0.89 PARP1 (0.75) PARP1PARP2
SCHEMBL19200089 0.89 PARP1 (0.62) PARP1PARP2
SCHEMBL19199910 0.88 PARP1 (0.79) PARP1PARP2
SCHEMBL19199983 0.87 PARP1 (0.80) PARP1PARP2
SCHEMBL12822197 0.87 PARP1 (0.76) PARP1PARP2
SCHEMBL22420900 0.87 PARP1 (0.74) PARP1PARP2
SCHEMBL15449622 0.87 PARP1 (0.77) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110088098-B Quinazolinone PARP-1 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-04-15 CN disclosed
WO-2017128036-A1 QUINAZOLINONE PARP-1 INHIBITOR AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE THEREOF 中国医学科学院药物研究所 2017-08-03 WO disclosed