SCHEMBL19200089

SCHEMBL19200089

O=C(c1cc(Cn2c(=O)[nH]c(=O)c3c(F)cccc32)ccc1F)N1CCN(CC(F)(F)F)CC1

nearest known ligand 0.62

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.62
PARP2 Q9UGN5 19/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19199863 0.89 PARP1 (0.79) PARP1PARP2
SCHEMBL30428242 0.86 PARP1 (0.61) PARP1PARP2
SCHEMBL12822554 0.86 PARP1 (0.61) PARP1PARP2
SCHEMBL29722305 0.85 PARP1 (0.63) PARP1PARP2
SCHEMBL15420832 0.85 PARP1 (0.63) PARP1PARP2
SCHEMBL30543559 0.85 PARP1 (0.56) PARP1PARP2
SCHEMBL12821953 0.85 PARP1 (0.56) PARP1PARP2
SCHEMBL12822239 0.85 PARP1 (0.61) PARP1PARP2
SCHEMBL29722477 0.85 PARP1 (0.65) PARP1PARP2
SCHEMBL12822603 0.85 PARP1 (0.65) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110088098-B Quinazolinone PARP-1 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-04-15 CN disclosed
WO-2017128036-A1 QUINAZOLINONE PARP-1 INHIBITOR AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE THEREOF 中国医学科学院药物研究所 2017-08-03 WO disclosed