SCHEMBL19200482

SCHEMBL19200482

NC1c2ccccc2C[C@@H]1NC(=O)C(c1ccc(F)cc1F)N1CCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 2/20 0.39
OXTR P30559 8/20 0.39
CYP3A4 P08684 2/20 0.39
AVPR2 P30518 2/20 0.39
AVPR1A P37288 2/20 0.39
NPY2R P49146 1/20 0.35
TSHR P16473 1/20 0.34
PYGL P06737 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
GHSR Q92847 1/20 0.33
MAPK14 Q16539 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33
OPRM1 P35372 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19182798 1.00 GRM7 (0.39) GRM7OXTRCYP3A4AVPR2AVPR1A
SCHEMBL19200400 0.89 GRM7 (0.41) GRM7OXTRCYP3A4AVPR2AVPR1A
SCHEMBL19200271 0.89 GRM7 (0.41) GRM7OXTRCYP3A4AVPR2AVPR1A
SCHEMBL19183412 0.89 GRM7 (0.41) GRM7OXTRCYP3A4AVPR2AVPR1A
SCHEMBL19200313 0.87 OXTR (0.40) GRM7OXTRCYP3A4AVPR2AVPR1A
SCHEMBL19182901 0.86 GRM7 (0.40) GRM7OXTRCYP3A4AVPR2AVPR1A
SCHEMBL19200515 0.86 GRM7 (0.40) GRM7OXTRCYP3A4AVPR2AVPR1A
Formic Acid SCHEMBL20678734 0.86 GRM7 (0.38) GRM7OXTRCYP3A4AVPR2AVPR1A
SCHEMBL19183402 0.85 GRM7 (0.36) GRM7OXTRCYP3A4AVPR2AVPR1A
SCHEMBL19183501 0.85 GRM7 (0.52) GRM7OXTRCYP3A4AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017131221-A1 INDANE DERIVATIVES AS MGLUR7 MODULATORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-03 WO disclosed