SCHEMBL1920462

SCHEMBL1920462

C=C(CCc1ccccc1C)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTBP2 P56545 1/20 0.47
ALDH1A1 P00352 2/20 0.46
TAAR1 Q96RJ0 1/20 0.46
NOTUM Q6P988 1/20 0.44
HPGD P15428 2/20 0.44
HTT P42858 2/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
LMNA P02545 2/20 0.40
PTGER1 P34995 1/20 0.40
PTGER4 P35408 1/20 0.40
PTGER3 P43115 1/20 0.40
PTGER2 P43116 1/20 0.40
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
CYP4F2 P78329 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL678766 0.90 CTBP2 (0.45) CTBP2ALDH1A1TAAR1NOTUMHPGD
SCHEMBL11399078 0.86 POLB (0.40) CTBP2ALDH1A1NPSR1PTGER1PTGER4
SCHEMBL7058525 0.81 CTBP2 (0.50) CTBP2ALDH1A1TAAR1NOTUMHPGD
SCHEMBL7441996 0.81 CTBP2 (0.59) CTBP2ALDH1A1HPGDHTTGAA
SCHEMBL28167993 0.81 NOTUM (0.45) ALDH1A1TAAR1NOTUMHPGDHTT
SCHEMBL323867 0.81 NPSR1 (0.61) CTBP2ALDH1A1TAAR1NOTUMHPGD
SCHEMBL29843936 0.81 NPSR1 (0.61) CTBP2ALDH1A1TAAR1NOTUMHPGD
SCHEMBL17940787 0.81 HTR2A (0.50) ALDH1A1PTGER1PTGER4PTGER3PTGER2
SCHEMBL1137802 0.80 AKR1B1 (0.52) TAAR1
Water SCHEMBL10936872 0.79 NPSR1 (0.59) CTBP2ALDH1A1TAAR1NOTUMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4121802-B1 HIGH REFRACTIVE INDEX SILOXANE INSERT MATERIALS FOR EMBEDDED CONTACT LENSES ALCON INC (CH) 2024-07-17 EP claimed
EP-3728339-B1 COMPOSITION FOR OPHTHALMOLOGICAL PRODUCTS AMO Ireland (IE) 2022-07-06 EP claimed
EP-2303331-B1 OPHTHALMIC DEVICE HAVING THERAPEUTIC AGENT DELIVERY CAPABILITY AND METHOD OF FORMING SAME ALCON INC (CH) 2022-01-26 EP claimed
EP-3200840-B1 LOW-WATER CONTENT ACRYLATE-ACRYLAMIDE COPOLYMERS FOR OPHTHALMIC DEVICES ALCON INC (CH) 2021-11-17 EP claimed
EP-3200839-B1 HYDROPHOBIC ACRYLATE-ACRYLAMIDE COPOLYMERS FOR OPHTHALMIC DEVICES NOVARTIS AG (CH) 2019-09-04 EP claimed
EP-3223870-B1 WET-PACK INTRAOCULAR LENS MATERIALS WITH HIGH REFRACTIVE INDEX NOVARTIS AG (CH) 2018-09-26 EP claimed
EP-3077016-B1 SOFT ACRYLIC MATERIALS WITH HIGH REFRACTIVE INDEX AND MINIMIZED GLISTENING NOVARTIS AG (CH) 2018-05-16 EP claimed
EP-2292672-B1 Biocompatible polymers and co-polymers comprising amino acids in the side chain CIS PHARMA AG (CH) 2018-05-09 EP claimed
EP-1888660-B1 BIOCOMPATIBLE POLYMERS AND CO-POLYMERS COMPRISING AMINO ACIDS IN THE SIDE CHAIN CIS PHARMA AG (CH) 2017-05-17 EP claimed
EP-2906970-B1 HIGH REFRACTIVE INDEX OPHTHALMIC DEVICE MATERIALS WITH REDUCED TACK NOVARTIS AG (CH) 2016-11-23 EP claimed
EP-2582409-B1 HIGH REFRACTIVE INDEX, ACRYLIC OPHTHALMIC DEVICE MATERIALS WITH REDUCED GLISTENINGS NOVARTIS AG (CH) 2014-09-10 EP claimed
EP-2225325-B1 HIGH REFRACTIVE INDEX OPHTHALMIC DEVICE MATERIALS ALCON INC (CH) 2011-06-01 EP claimed
EP-1080382-B1 HIGH REFRACTIVE INDEX OPHTHALMIC DEVICE MATERIALS ALCON INC (CH) 2009-07-08 EP claimed
EP-1080381-B1 HIGH REFRACTIVE INDEX OPHTHALMIC DEVICE MATERIALS PREPARED USING A POST-POLYMERIZATION CROSS-LINKING METHOD ALCON MFG LTD (US) 2005-07-27 EP claimed
EP-1002244-B1 METHOD OF PREPARING FOLDABLE HIGH REFRACTIVE INDEX ACRYLIC OPHTHALMIC DEVICE MATERIALS ALCON LAB INC (US) 2003-02-26 EP claimed
EP-1079870-B1 BICOMPOSITE INTRAOCULAR LENS AND METHOD FOR ITS PREPARATION ALCON LAB INC (US) 2001-11-14 EP claimed
EP-1071482-B1 INTRAOCULAR LENS COATING COMPOSITIONS ALCON LAB INC (US) 2001-10-04 EP claimed
US-4284707-A Photocurable light-sensitive composition SOMAR MANUFACTURING CO., LTD. (JP) 1981-08-18 US claimed
EP-3728339-B1 COMPOSITION FOR OPHTHALMOLOGICAL PRODUCTS AMO Ireland (IE) 2022-07-06 EP disclosed
US-4284707-A Photocurable light-sensitive composition SOMAR MANUFACTURING CO., LTD. (JP) 1981-08-18 US disclosed