SCHEMBL1920505

SCHEMBL1920505

COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OC1CCN(C(=O)N2CCCCC2)CC1.COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OC1CCN(CC(N)=O)CC1

nearest known ligand 0.75

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 9/20 0.75
EGFR P00533 15/20 0.70
ERBB4 Q15303 2/20 0.58
GAK O14976 1/20 0.58
RIPK2 O43353 1/20 0.58
NR1I2 O75469 1/20 0.58
LCK P06239 1/20 0.58
ADORA3 P0DMS8 1/20 0.58
CHRM1 P11229 1/20 0.58
SRC P12931 1/20 0.58
DRD2 P14416 1/20 0.58
ADRA2C P18825 1/20 0.58
SLC6A2 P23975 1/20 0.58
MC3R P41968 1/20 0.58
JAK3 P52333 1/20 0.58
SLC6A3 Q01959 1/20 0.58
PDE4D Q08499 1/20 0.58
KCNH2 Q12809 1/20 0.58
RIPK3 Q9Y572 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29623469 0.94 ERBB2 (0.84) ERBB2EGFRGAKRIPK2RIPK3
SCHEMBL185530 0.94 ERBB2 (0.84) ERBB2EGFRGAKRIPK2RIPK3
SCHEMBL185050 0.93 EGFR (0.77) ERBB2EGFR
SCHEMBL29623692 0.93 EGFR (0.77) ERBB2EGFR
SCHEMBL1447161 0.92 EGFR (0.78) ERBB2EGFR
SCHEMBL4879883 0.90 ERBB2 (0.81) ERBB2EGFRGAKRIPK2RIPK3
SCHEMBL12743511 0.87 FBP1 (0.65) ERBB2EGFRERBB4
SCHEMBL24637510 0.87 ERBB2 (0.86) ERBB2EGFRGAKRIPK2RIPK3
SCHEMBL12743207 0.87 EGFR (0.79) ERBB2EGFR
SCHEMBL12743515 0.87 EGFR (0.68) ERBB2EGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2326374-A1 INHALER Boehringer Ingelheim International GmbH (DE) 2011-06-01 EP disclosed
WO-2009153049-A1 INHALER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-12-23 WO disclosed